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3-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
4-benzyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-1-(3-methylphenyl)-4-(quinoxaline-5-carbonyl)piperazin-2-one
N'1-[(3R,4S)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
4-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridin-1-ium-1-olate
3-(1-hydroxyhexan-2-yl)-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(pyrrolidin-3-yl)acetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(3-methylpiperidin-1-yl)propanamide
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-4-fluorobenzamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
4-[(4-tert-butylphenyl)methyl]-N-(6-cyanopyridin-3-yl)piperazine-1-carboxamide
N-{1-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperidin-4-yl}acetamide
2-(2-hydroxyethyl)-9-(2-oxoimidazolidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3-methylbenzoyl)piperidine
2-{9-[(5-methylthiophen-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(2R,6R)-4-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
[(3R,4S)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2,6-dimethoxy-N-[2-(4-methylmorpholin-2-yl)ethyl]pyridine-3-carboxamide
1-[4-methyl-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]pyrrolidin-2-one
2-{4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]piperidin-1-yl}acetic acid
N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(3,4-difluorophenyl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[(2-fluorophenyl)methyl]acetamide
1-(2-{1-[2-(2,5-dimethylphenyl)acetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2-chlorophenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
3-[1-(1H-1,2,4-triazol-5-yl)ethyl]-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-2-carboxamide
N-ethyl-N-[2-(morpholin-4-yl)ethyl]piperidin-3-amine
5-ethyl-2-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]pyridine
(3S,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-propylpyrrolidine-3-carboxylic acid
6-{4-[1-(2-methoxyacetyl)piperidine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
4-{3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}morpholine-2-carboxylic acid
7-(3,5-dichloro-2-methoxybenzoyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-methylbut-2-en-1-one
N-[2-(2-ethoxyphenoxy)ethyl]-N,1-dimethyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
ethyl 1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2,5-dimethylpyrimidine
1-(3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
N-(2,3-dihydro-1H-inden-4-yl)-4-(1,3-dihydroxypropan-2-yl)morpholine-2-carboxamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
(3S,5R,9R)-11-(3,5-dichlorobenzoyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyloxolane-2-carboxamide
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dimethylpyridine
7-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one