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4-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)azetidin-3-yl]pyridine
7-[(4-fluorophenyl)methyl]-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
7-(2,3-dihydro-1-benzofuran-7-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)azetidin-3-ol
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-(methoxymethyl)piperidine
2-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-3,4-dimethoxypyridine
2-phenoxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-[({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]-N-methylfuran-2-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2H-1,3-benzodioxol-5-yloxy)ethan-1-one
N-[(3R,4S)-4-(propan-2-yl)-1-(4,4,4-trifluorobutyl)pyrrolidin-3-yl]furan-3-carboxamide
(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazol-4-yl)methanol
2-methyl-3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
6-(1,4-dioxan-2-ylmethyl)-5,6-dihydro-1,6-naphthyridin-5-one
2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(3S,5S)-5-[1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1-methylpyrrolidin-3-amine
(1R,3S)-7-(6-chloro-2H-chromene-3-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-2-[3-(trifluoromethyl)phenyl]acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(4-methyloxan-4-yl)methyl]acetamide
1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
2-{2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-6-methoxyphenoxy}propanoic acid
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(8-methoxyquinolin-5-yl)methyl](methyl)amino}acetamide
4-[5-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
2-(1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)ethan-1-ol
(1S,4S)-2-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-2-azabicyclo[2.2.1]heptane
N-[(2S,4R,6S)-2-(4-acetamidophenyl)-6-(2-phenylethyl)oxan-4-yl]acetamide
(4S)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenyl-1,3-oxazolidin-2-one
N-[(4-fluorophenyl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
7-(2-methoxyethyl)-2-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
6-{[4-(4-methoxyphenyl)butan-2-yl]amino}-2-methylheptan-2-ol
ethyl 4-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
N-[4-(5-tert-butyl-1H-pyrazol-3-yl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
1'-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(1S,5R)-6-benzyl-3-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-cycloheptanecarbonyl-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-5-phenyl-1,2-oxazole-3-carboxamide
4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-ethylpyrimidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
7-methyl-3-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]-1H-indole
1-(2,5-dimethoxyphenyl)-2-(2,2-dimethyloxan-4-yl)-1H-imidazole
(4aS,8aR)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(3S,4R)-4-(pyridin-3-yl)-1-[1-(pyrrolidin-1-yl)cyclohexanecarbonyl]pyrrolidine-3-carboxylic acid
2-{[(3-ethoxyphenyl)methyl](quinolin-3-ylmethyl)amino}ethan-1-ol
4-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-1-(2-phenylphenyl)piperazin-2-one
2-methyl-1-[1-(4-methyl-1H-imidazole-5-carbonyl)azetidin-3-yl]piperidine
1'-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)spiro[indene-1,4'-piperidine]
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide