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2-(2-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
N-[1-(pyridin-3-yl)propan-2-yl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(2-oxoazepan-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(1,3-benzothiazol-2-yl)-4-(2-methoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}(ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
ethyl 5-(dimethyl-1,2-oxazole-4-carbonyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(3-methoxyphenyl)-3-{1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}propanamide
6-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-N-ethylpyridine-3-carboxamide
2-(2,3-difluorophenyl)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
N-(oxolan-3-yl)-4-[(3-oxopiperazin-1-yl)sulfonyl]benzamide
2-{2-[4-(3-fluorophenoxy)piperidin-1-yl]ethyl}pyridine
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(methoxymethyl)-1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
8-methoxy-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}quinoline
1-(oxan-4-yl)-4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]piperazine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-[9-(4-ethoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
2-[(2-fluorophenyl)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
3-{2H,4H,5H,6H-cyclopenta[c]pyrazol-2-yl}-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-ethylpiperidine-1-carboxamide
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(piperidin-3-yl)benzamide
5-methyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}thieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-3-yl}benzoic acid
3-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
methyl 5-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]carbamoyl}-1-methyl-1H-pyrazole-3-carboxylate
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-ol
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(4-methylbenzoyl)piperidine
6-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-benzyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}propanamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 3-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]propanoate
1-ethyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-[4-(thiophene-2-carbonyl)morpholin-3-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
N-(cyclohexylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3R,5S)-5-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-3-ol
(3R,4R)-4-amino-1-(7,8-dimethylquinolin-4-yl)piperidin-3-ol
6-(1,3-benzothiazol-2-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}-N-[2-(1H-pyrazol-1-yl)ethyl]pyridine-3-carboxamide
1-(3-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)piperidine-4-carboxamide
N-[4-methyl-3-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)phenyl]propanamide
2-(3-fluorophenyl)-N-({7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-[(3R,4S)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-3-(2-methylphenyl)propanamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethylpropanamide
(3S,4R)-N-(5-chloro-2-methoxyphenyl)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carboxamide