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2-methyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1H-1,3-benzodiazole-5-carboxamide
3-(2-fluorophenyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
(2S)-2-amino-2-phenyl-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,N-diethyl-5-methyl-1H-pyrazole-4-carboxamide
(2S)-2-amino-1-[4-(3-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(3-methoxypropyl)benzamide
2-ethoxy-4-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
2-(2-chloro-4-fluorophenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
N-(1H-1,3-benzodiazol-5-yl)-4-[(oxolan-3-yl)sulfamoyl]benzamide
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methanol
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-methyl-4-(5-methyl-2-phenylfuran-3-carbonyl)-1,4,9-triazaspiro[5.5]undecane
methyl 3-[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]propanoate
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
5-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1-benzothiophene-5-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1,4-dioxane-2-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)spiro[azepane-4,2'-chromene]
N-{2-oxo-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1,2,3,4-tetrahydroquinolin-7-yl}methanesulfonamide
N-[(2S,4R,6S)-2-(2-phenylethyl)-6-(quinoxalin-2-yl)oxan-4-yl]acetamide
1-(1H-imidazol-2-ylmethyl)-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid
6-(pyrrolidin-1-ylmethyl)-4-[4-(trifluoromethyl)benzoyl]-1,4-oxazepan-6-ol
(4aS,8aR)-6-(2,6-difluorobenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
7-[2-(3-methoxyphenoxy)ethyl]pyrazolo[1,5-a]pyridine
3-{[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]methyl}-N,N-dimethylbenzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-[1-(2,6-dimethylquinoline-3-carbonyl)piperidin-4-yl]-2-methylpropan-1-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-(2,2-diphenylethyl)-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(methylsulfanyl)-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]ethan-1-one
4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)morpholine
5-{[2-(diethylamino)ethyl]amino}-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 1-[(3R,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{2-oxo-2-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
(8R,9aS)-8-hydroxy-2-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
1-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
(3R,4R)-1-(naphthalen-2-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
(3S,5R,9R)-11-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
7-chloro-1-methyl-N-[2-(morpholin-4-yl)butyl]-1H-indole-2-carboxamide
2-ethoxy-5-{2-[(1-propanoylpiperidin-4-yl)amino]pyrimidin-4-yl}benzoic acid
6-methyl-2-[(2-methylphenyl)methyl]-1-(pyridin-2-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
ethyl 3-benzyl-1-[(2,5-dimethoxyphenyl)carbamoyl]piperidine-3-carboxylate
(4aR,7aS)-1-(2-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[(5-methylpyrazin-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-chloro-N-(2-methoxyethyl)-4-({1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}oxy)benzamide