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N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]oxolane-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-1H-1,3-benzodiazol-2-yl)methyl](oxolan-2-ylmethyl)amine
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1-(pyrimidin-2-yl)piperidine-4-carboxamide
1-[(2,4-difluorophenyl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(oxolan-3-ylmethyl)piperidin-4-yl]acetate
4-(2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)morpholine
2-(4-methoxyphenyl)-4-{4-[4-(2-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridazine
(2S)-N-[1-benzyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(methylamino)propanamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
5-{[benzyl(methyl)amino]methyl}-N-cycloheptyl-N-ethyl-1,2-oxazole-3-carboxamide
N5-[(1-ethylpiperidin-3-yl)methyl]-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
(4aR,8aR)-1-[4-(4-methylpiperazin-1-yl)benzoyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine
6-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
5-(4-methoxy-3,5-dimethylphenyl)pyridine-3-carboxamide
5-{[3-phenyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
methyl 1-ethoxy-2-oxo-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 2-[3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenylpropanamido]acetate
1-methyl-5-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-2-one
N-(2-fluorophenyl)-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
ethyl 4-{[1-(pyrrolidine-1-carbonyl)azepan-3-yl]amino}piperidine-1-carboxylate
3-(5-{3-[(dimethylamino)methyl]-4-methoxyphenyl}-4-phenyl-1H-imidazol-1-yl)propan-1-ol
2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}benzonitrile
(2S)-2-amino-2-cyclohexyl-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
5-[(dimethylamino)methyl]-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]furan-2-carboxamide
8-(3-aminopropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4,6-dimethyl-13-[2-(morpholin-4-yl)pyridin-3-yl]-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
N2,N2-dimethyl-N5-[(2-methylpyrimidin-5-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-5-phenylpentane-1,5-dione
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(pyridin-2-ylsulfanyl)acetamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amine
N-{1-oxo-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-2-yl}methanesulfonamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-(3,4-dimethoxybenzoyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
(4aS,7aR)-1-(morpholine-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclobutanecarbonyl-N-[2-(5-methylfuran-2-yl)ethyl]piperidine-4-carboxamide
(4aR,8aR)-2-(1H-imidazol-2-ylmethyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
3-fluoro-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(3-methoxypropyl)-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(4aS,8aR)-6-(isoquinolin-1-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
2-(5-acetylthiophen-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
2-methyl-6-(piperidin-4-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-4-amine
1-[5-(cyclopropylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
2-(3-{[(2-methoxyethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[(1-benzylpiperidin-4-yl)methyl]-N,4-dimethyl-1,3-thiazol-2-amine
N-[(2,5-difluorophenyl)methyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide