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5-(ethoxymethyl)-1-[(4-ethylphenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-(5-cyclopentaneamido-2-methylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
N-cycloheptyl-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2-{2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
(2-methoxyethyl)({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
N-[(3R,4S)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-propylpyrrolidin-3-yl]-2-methoxyacetamide
4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
1-{2-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(3S,4S)-1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
3-(3-acetamidophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
(3S,7S,8aS)-7-{[(3-fluoro-4-methylphenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(dimethylamino)-2-(4-fluorophenyl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-(1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-yl)acetamide
(4aR,8aS)-N,N-dimethyl-1-(3-phenylprop-2-ynoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
4-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
1-(2-chlorophenyl)-3-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}urea
2-ethyl-9-[2-(2,3,4-trifluorophenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzonitrile
(4S)-4-amino-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butanoic acid
(3R,5S)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(1H-indol-4-ylmethyl)(methyl)(1H-pyrazol-3-ylmethyl)amine
(3S)-4-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-{[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
[3-(azepan-1-yl)propyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
1-[1'-(4,6-dimethylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
ethyl[(5-ethylpyridin-2-yl)methyl][(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-methyl-2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}aniline
2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-cyclopentyl-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(2R,3R,6R)-5-[(4-methoxy-3-methylphenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
4-(1-methyl-1H-imidazol-2-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[2-(4-methylphenoxy)ethyl]pyridin-2-amine
N-[3-(3-fluorophenyl)phenyl]-1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}benzamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(4-{4-[(1,4-dioxan-2-ylmethyl)(methyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
1-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-1-(propan-2-yl)-3-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
N'-cyclopentyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}butanediamide
2-benzyl-8-(4-fluoro-3-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-ol
1-[(4-chlorophenyl)methyl]-N-methyl-N-(pyrimidin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide