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1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
4-{furo[3,2-c]pyridin-4-yl}-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
2-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
3-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2,5-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1,3-thiazole-4-carboxamide
2-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-8-methyl-2,8-diazaspiro[4.5]decan-3-one
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-({[(3R,4R)-1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6,8-dioxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.4]nonane-2-carboxamide
2-(4-{1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
N-(2-oxooxolan-3-yl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
diethyl({[3-(2-methylpyrrolidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
4-(4-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
1-(6-methylpyridin-2-yl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
4-(2-chlorobenzenesulfonyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-{[4-(cyclooctyloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
4-[(dimethylamino)methyl]-1-[3-(4-fluorophenoxy)propyl]azepan-4-ol
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
1-methyl-1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-[1-(furan-2-yl)ethyl]-N-methyl-2-[(thiophen-2-ylmethyl)amino]benzamide
N-[(3-methyl-7-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]furan-2-carboxamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-4-(morpholin-4-yl)benzamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-methyl-1-{[3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxamide
5-phenyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-6-[(3-ethoxy-4-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-2-methyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
5-(4-fluorophenyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[(2-methoxyethyl)sulfamoyl]-5-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]benzoic acid
4-[(3-chlorophenyl)methyl]-1-(furan-3-ylmethyl)-1,4-diazepan-5-one
8-cyclobutanecarbonyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclobutanecarboxamide
N-(1-phenyl-1H-pyrazol-5-yl)-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
3-[(5-fluoroquinazolin-4-yl)amino]piperidin-2-one
5-(4-acetyl-2-methoxyphenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
4-chloro-N,1,5-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
3-{1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}benzoic acid
5-[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
1-cyclopropyl-N-[3-(1H-imidazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
[(2,3-difluoro-6-methoxyphenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
N-[2-({2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-4-fluorobenzamide