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1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
5-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(5-methyl-1H-imidazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
4-{5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(3-ethoxyphenyl)pyridine-2-carbonitrile
4-{1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]azetidin-3-yl}pyridine
1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-methoxypropan-2-yl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
3-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
5-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}thiophene-2-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-6-methyl-2-propylpyrimidin-4-amine
4-methoxy-N-{[1-(thiophene-3-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
4-(2-ethoxyphenyl)-6-methylpyrimidin-2-amine
4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetamide
4-(4-chlorophenyl)-1-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}piperidin-4-ol
N-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-2-(pyridin-2-yl)piperidine-1-carboxamide
4-methyl-5-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrimidin-2-amine
2-cyclopropyl-8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
6-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,3-dihydro-1-benzofuran-5-carboxamide
N-[(3S,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
5-[7-(3-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N-methylfuran-2-carboxamide
2-(3,4-dichlorophenyl)-4-(3-fluoro-2-methoxybenzoyl)morpholine
N-[2-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-propyl-2,8-diazaspiro[4.5]decan-3-one
1-{2-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-pyrrole
N-({5-[(3-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-(2-{methyl[(3-methylthiophen-2-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
N-ethyl-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)pyrimidin-4-amine
(1S,4S)-2-(2-chlorophenyl)-5-[1-(2-phenylethyl)piperidin-4-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
[(3-methoxyphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-(2-hydroxyethyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-tert-butyl-6-(2,3-dichlorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-(5-{6-amino-5-cyano-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridin-2-yl}thiophen-3-yl)acetic acid
4-{1-[(1S)-2,3-dihydro-1H-inden-1-yl]-1H-imidazol-2-yl}pyridine
(3R,4R)-4-amino-1-({3-[(4-chlorophenyl)methoxy]phenyl}methyl)piperidin-3-ol
2-[3-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-cyclopentyl-4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[4-(4-phenylpyrimidin-2-yl)piperazin-1-yl]-2-(pyrrolidin-3-yl)ethan-1-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(3-methylpiperidin-1-yl)acetamide
5,7-dimethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide