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1-ethyl-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
(3aS,6aS)-2-(naphthalene-1-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(diethylamino)ethyl]-N-ethyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-benzyl-N-methyl-N-[2-(pyridin-4-yl)ethyl]piperidine-2-carboxamide
5-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
(3aR,6aR)-2-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
5-{[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-N-methylfuran-2-carboxamide
N-[(2S,4R,6R)-2-[2-(benzylamino)pyrimidin-5-yl]-6-(propan-2-yl)oxan-4-yl]acetamide
methyl 2-{8-[(2-chloro-6-fluorophenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-(quinolin-8-ylmethyl)propanamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-[3-(furan-2-yl)-1H-pyrazol-5-yl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]thian-4-amine
(3aS,6aS)-2-[2-(2-chloro-6-fluorophenyl)acetyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(3-fluoro-4-methoxyphenyl)-3-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
5-(propan-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanamide
2,2-diphenyl-1-[4-(1,2,5-thiadiazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
2-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
1-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}azepane
2-benzyl-5-(4-cyclohexylpiperazine-1-carbonyl)-1,3-benzoxazole
(2R,6S)-4-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-2,6-dimethylmorpholine
N-methyl-N-(1-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
2-(4-methoxy-3-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-amino-4-(1,3-dimethyl-1H-pyrazol-4-yl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
3-methanesulfonyl-N-[(3R,4S)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
5-methyl-3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-indazole
6-fluoro-2-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2-dihydroquinoline-4-carboxamide
4-chloro-2-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]phenol
1-{1-[(2-ethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
3-(3-fluorophenyl)-6-(1H-indole-6-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)methyl]piperidine
N-[2-(4-methoxyphenyl)propan-2-yl]-1-methyl-1H-imidazole-5-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(dimethylamino)pentyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
1-{2-[3-(2-chlorophenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
N-({7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-benzyl-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-sulfonamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(2-methoxyphenoxy)piperidine
4-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamido]oxane-4-carboxylic acid
3-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(5-methanesulfonamido-2-methylphenyl)urea
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{9-oxa-2-azaspiro[5.5]undecan-2-yl}butan-1-one
N-[1-({[2-(2-methyl-1-phenyl-1H-indol-3-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide