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2-methoxy-N-{[5-(quinolin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-[(3R,4R)-3-hydroxy-1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl]pyridine-2-carboxamide
4-{1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
4-(dimethyl-1,2-oxazol-4-yl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]ethyl}morpholine
3-[1-(6-fluoro-4-methylquinolin-2-yl)piperidin-3-yl]-N,N-dimethylpropanamide
4-[2-(hydroxymethyl)piperidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
5-{[(4aS,7aR)-4-(3-methylbut-2-en-1-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-2-hydroxybenzoic acid
2-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]pyridine-4-carbonitrile
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-[4-(ethoxymethyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(pyridin-4-yl)propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
2-[(4aR,7aS)-6,6-dioxo-4-[2-(2-oxopyrrolidin-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
4,6-dimethyl-1-[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethyl]-1,2-dihydropyrimidin-2-one
7-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-[3-(carbamoylmethoxy)phenyl]-N,N-bis(propan-2-yl)benzamide
2-(2-hydroxyethyl)-6-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
6-[1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
3-ethoxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
(4aS,7aR)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,5-dimethyl-1H-pyrazole
(1R,3S)-7-{[4-(2-methylpropyl)phenyl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}oxolane-3-carboxamide
2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
(1S,5R)-3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2,6-dioxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
7-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 5-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
6-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
4-{5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}phenol
2-(pyridin-3-ylmethyl)-9-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
ethyl 4-[6-(thian-4-yl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
1-(carbamoylmethyl)-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)piperidine-4-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{5-[1-(2-methoxyethyl)pyrrolidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridazine
7-(2-cyclohexylethyl)-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(2,4-difluorophenyl)-1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
3-(1-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-N-(2-phenylethyl)formamido)propanamide
1-(1-propanoylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide