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N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[(3-methoxyphenyl)methyl]piperidine
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-chloro-4-fluorophenyl)ethan-1-one
methyl(quinolin-6-ylmethyl)[(3-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
9-(3-chloro-4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-5-(1,2,3,4-tetrahydronaphthalen-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{1-azabicyclo[2.2.2]octan-3-yl}-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
1-tert-butyl-N-(2,3-dihydro-1H-inden-2-yl)-5-oxo-N-propylpyrrolidine-3-carboxamide
1-(2-oxo-2-{4-[(pyridin-2-yl)amino]piperidin-1-yl}ethyl)piperidine-4-carboxamide
5-(dimethylamino)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,3-dihydropyridazin-3-one
6-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
5-methyl-2-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-1,3-benzoxazole
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
7-cyclohexyl-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(pyrimidin-4-ylmethyl)-1,3-oxazole-4-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
3-ethyl-8-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-({ethyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)-2-hydroxybenzoic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(quinazolin-4-yloxy)acetamide
[3-(cyclopropylmethyl)-1-(4-propylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
1-ethyl-4-{1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}piperazine
4-(dimethylsulfamoyl)-N-[3-(pyridin-2-yl)phenyl]piperazine-1-carboxamide
N-methyl-2,6-dioxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
4-[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]-4H-1,2,4-triazole
2-(4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
(4aS,8aR)-6-(2-aminopyridine-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
4-ethyl-2-methyl-6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-phenoxypiperidine-4-carboxylic acid
(2S,4R)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
N-[(3S,4R)-4-(propan-2-yl)-1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]acetamide
N-(3-fluorophenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-({3-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)-1H-pyrazole
N-methyl-N-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}cyclohexanamine
(butan-2-yl)(3-phenylprop-2-yn-1-yl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
4-(2-fluoro-5-methylphenoxy)-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxylic acid
1-(2-ethoxyphenyl)-4-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
7,7-dimethyl-2-[1-(2-methylpropyl)pyrrolidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2-fluorophenyl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-[(2-phenoxypyridin-3-yl)methyl]-1-phenylcyclopropane-1-carboxamide
4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-chloro-3-methoxyphenyl)-4-(oxolane-2-carbonyl)-1,4-diazepane-1-carboxamide
(3S,4R)-1-(4-oxo-4H-chromene-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid