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5-acetyl-N-ethyl-2,4-dimethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrrole-3-carboxamide
4-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)pyrimidine
2-(4-fluorophenyl)-2-hydroxy-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-2-carbonitrile
3-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
7-(cyclohexylmethyl)-2-(4,4,4-trifluorobutanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-cyclopentyl-1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1H-1,2,3-triazole-5-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2,3,4-trimethoxybenzamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[4-(hydroxymethyl)benzoyl]piperidin-4-yl]pyridine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
ethyl 1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-4-carboxylate
2-{1-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1H-imidazol-2-yl}pyridine
1-ethyl-3,5-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
N-[1-(2,4-difluorophenyl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
7-(cyclopropylmethyl)-2-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-(6-methylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-[(5-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
N-{1-[(5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]pyrrolidin-3-yl}acetamide
methyl 3-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoate
N-cyclopentyl-4-(4-{[2-(3-fluorophenyl)ethyl]amino}piperidin-1-yl)benzamide
2-(2-{[2-(dimethylsulfamoyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
3-{5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-yl]-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(1S,5R)-3-[(1-methyl-1H-indol-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-6-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,6-dihydropyridazine-3-carboxamide
N-methyl-6-oxo-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-[5-(methoxymethyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
4-fluoro-N-[3-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)phenyl]benzene-1-sulfonamide
2-(1-methyl-1H-indol-3-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
3-[2-(3,4-difluorophenyl)ethyl]-1-(1H-imidazol-4-ylmethyl)piperidine
3-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
(2R)-2-amino-N,4-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pentanamide
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methylphenol
N-cyclopropyl-6-(4-methoxyphenyl)-7-methyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[(1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
3-ethyl-1-(3-methylbutyl)-8-{[4-(trifluoromethoxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
5-[5-(1-cyclobutanecarbonylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
(5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}furan-2-yl)methanol
5-cyclopropyl-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazole
5-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(3-methylbut-2-en-1-yl)-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
2-cyclopropanecarbonyl-8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[(8-methoxyquinolin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[(2,3-dihydroxypropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide