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3-({[(dimethyl-1,2-oxazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
(5S,9aS,9bS)-5-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(1,2-oxazol-3-ylmethyl)benzamide
2-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}benzoic acid
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-methylbenzamide
{3-[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
3-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
2,6-dimethoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyridine-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)(quinolin-2-ylmethyl)amine
1-(2-methoxy-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
({4-ethyl-5-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-[2-(2,3-dimethylphenoxy)ethyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
1-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
1-{2-[4-(2-ethylphenyl)piperazin-1-yl]-2-oxoethyl}imidazolidin-2-one
4-{[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-{[2-(pyridin-3-yloxy)propyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[4-(ethylcarbamoyl)phenyl]-4-(6-ethylpyrimidin-4-yl)piperazine-1-carboxamide
(1S,6R)-N-[3-(3-chlorophenyl)phenyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1-[3-(methylsulfanyl)phenyl]urea
N,4-dimethyl-2-(propan-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazole-5-carboxamide
2-methoxy-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(quinolin-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-amino-8-(2-chloro-4-fluorophenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
7-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-5-[2-(piperidin-1-yl)ethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-methyl-2-(2-{[methyl(3-methylbutyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
5-fluoro-N-(1H-indol-4-ylmethyl)quinazolin-4-amine
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[(1-methoxypropan-2-yl)amino]methyl}-1,2-dihydroquinolin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(1H-pyrazol-4-yl)butanamide
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-(prop-2-en-1-yl)urea
4-(3-methylbutyl)-3-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)piperazin-2-one
7-(2-phenylethyl)-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1H-imidazol-4-ylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
(3S,4R)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methoxypiperidin-4-amine
3-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}benzonitrile
4-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}pyridine
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[4-(propan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
N-[(3S,4R)-1-(3-cyanobenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[(2-fluorophenyl)formamido]-N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)propanamide
5-{5-[2-(1H-indol-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-benzyl-N-methyl-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-amine
5-(4-acetylpiperazin-1-yl)-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4S)-4-[methyl({[3-(5-methylfuran-2-yl)phenyl]methyl})amino]oxolan-3-ol
1-{2-methyl-1-[3-(4-methylphenoxy)azetidin-1-yl]propan-2-yl}piperidine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine