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2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
4-(1-{2-[ethyl(methyl)amino]-2-methylpropyl}-4-phenyl-1H-imidazol-5-yl)benzoic acid
1-(2-{1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2-fluoro-5-methoxyphenyl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
9-(6-ethyl-2-methylquinoline-4-carbonyl)-6-oxa-9-azaspiro[4.5]decane
N-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-propoxypiperidine-1-carboxamide
3-methyl-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-(thiophen-3-yl)acetic acid
1-ethyl-4,6-dimethyl-2-oxo-N-(2,2,2-trifluoroethyl)-1,2-dihydropyridine-3-carboxamide
5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclohexyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydroisoquinolin-1-one
3-(dimethylamino)-N-[3-methyl-1-(4-methylquinolin-2-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(4-methyl-1,4-diazepan-1-yl)propan-1-one
4-benzyl-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(3S,4R)-4-methoxyoxolan-3-yl]propanamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(5-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(hydroxymethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
(2S,4S,5R)-4-[cyclopropyl(ethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
N-(1-{4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}pyrrolidin-3-yl)acetamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-amino-4-{3-[(dimethylamino)methyl]-4-methoxyphenyl}-6-(1-methylcyclopropyl)pyridine-3-carbonitrile
N6-cyclopentyl-N5-ethyl-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}piperazine-1-sulfonamide
2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-ethyl-1,4-dimethyl-1H-pyrazol-5-amine
[(3R,4R)-1-(2-methoxypyridine-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(3-fluorophenyl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
3-methyl-4-({4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}methyl)pyridine
N6-cyclopropyl-N4-methyl-N4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidine-2,4,6-triamine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methylphenyl)propanamide
N3-methyl-1-(3-methylbutyl)-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
8-(4-amino-3-hydroxybutanoyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-imidazole
2-methoxy-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]butan-1-one
(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazol-2-yl)methanol
4-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
7-[2-(trifluoromethyl)morpholine-4-carbonyl]quinoline
1-(3-oxo-3-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
3-(2-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenyl-N-(propan-2-yl)propanamide
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
8-[4-(hydroxymethyl)benzoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-[2-(3,4-dimethylphenoxy)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
propan-2-yl N-[(3S,5S)-5-{[(5-fluoro-2-methylphenyl)methyl]carbamoyl}-1-methylpyrrolidin-3-yl]carbamate