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3-ethyl-4-(6-ethyl-2-methylquinoline-4-carbonyl)piperazin-2-one
1-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
(3R,4R)-3-cyclobutyl-1-(3-fluoropyridin-4-yl)-4-methylpyrrolidin-3-ol
(3S)-1-[2-amino-7-(pyrazine-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
N-[4-(3-fluorophenyl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
(1-methyl-1H-imidazol-2-yl)({1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl})methanol
1-methyl-N-(1,4-oxazepan-6-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
{[5-(1-cycloheptanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
2-(dimethylamino)-1-(3-hydroxyazetidin-1-yl)-2-(3-methylphenyl)ethan-1-one
(3aR,6aR)-2-(1-phenylcyclopentanecarbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{4-[(2-chlorophenyl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl}methanol
4-(cyclopropylmethyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl({[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})propylamine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
methyl 8-[(3-methylthiophen-2-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-[2-(2-chlorophenyl)-2-hydroxyacetyl]-1-(3-methoxyphenyl)piperazin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-cyclopentyl-N-methylacetamide
2-[(3-fluorophenyl)methyl]-4-(thiophene-2-sulfonyl)morpholine
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
1-(1-benzofuran-2-carbonyl)-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
(2S,4S)-4-amino-N-methyl-1-(1-phenylcyclopropanecarbonyl)pyrrolidine-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-propyl-1H-pyrazole-4-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-thiazole-5-carboxamide
[(2S,6S)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-ethyl-2-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
N,N-dimethyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
[3-(3-methoxypropyl)-1-(4-methylpiperidine-4-carbonyl)piperidin-3-yl]methanol
1-[(2-hydroxy-5-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-1,4-diazepane-6-carboxylic acid
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3-fluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-({5-[1-(cyclobutylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
[(3S,5R)-1-(1H-indazole-3-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
2,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}quinoxaline-6-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-(piperidin-1-ylmethyl)phenyl]urea
5-acetyl-2,4-dimethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrrole-3-carboxamide
1-cyclopentyl-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]butanamide
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
1-(2-methylpropyl)-5-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-hydroxypyridine-3-carboxamide