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2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(6-methylpyridazin-3-yl)piperazin-2-one
(3R)-1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-3,4,4-trimethylpyrrolidin-3-ol
(1R,2R,6S,7S)-4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
5-{2-[3-(benzyloxy)phenyl]-1H-imidazol-1-yl}-1-methylpiperidin-2-one
1-{[1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one
[(2E)-3-(furan-2-yl)prop-2-en-1-yl][(2-methoxyphenyl)methyl]propylamine
2-[(4aR,7aS)-6,6-dioxo-4-(piperidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-cyclopentyl-N-methyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
3-[5-(2-hydroxy-3-methylbutanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N,N-dimethyl-6-(3-{1-[(6-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazin-3-amine
4-fluoro-3-(2-phenylmorpholine-4-carbonyl)benzene-1-sulfonamide
N-[2-(3-methoxyphenyl)phenyl]-1-(6-methylpyrimidin-4-yl)piperidine-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(5-methylfuran-2-yl)benzamide
3-fluoro-4-methoxy-N-(1,2-oxazol-3-ylmethyl)benzamide
ethyl 5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-(2,5-dimethylfuran-3-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-3-hydroxy-2-{[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazol-5-yl]formamido}propanamide
3-[(3R,4S)-1-(3-fluoro-4-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(thiophen-2-yl)ethyl]benzamide
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(1H-pyrrol-1-yl)propanamide
N-(2-{1-[(2-chloro-5-fluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
methyl 4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)benzoate
2-(2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
(1S,4S)-2-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]diphenylmethanol
1-(2-hydroxyethyl)-5-(pyridine-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazol-2-yl)propan-1-ol
ethyl 7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
3-(2-chlorophenoxy)-1-[4-(difluoromethoxy)benzoyl]azetidine
9-methoxy-4-(4-methylbenzenesulfonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 4-[(7-chloro-2-ethyl-3-methyl-1-benzofuran-5-yl)carbamoyl]piperazine-1-carboxylate
2-(2-oxo-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-1-yl)benzonitrile
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3S,9aR)-3-benzyl-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(diphenylmethyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazine
(3S,4S)-4-(dimethylamino)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
1-(2-aminoethyl)-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
9-(5-methyl-1,2-oxazole-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methyl-1,4-diazepane
2-methyl-4-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)-6-propylpyrimidine
2-(6-ethyl-5-fluoropyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}carbamoyl)-2,1,3-benzoxadiazol-1-ium-1-olate
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidine-3-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propan-1-one
6-{[(4-methylphenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-N,N-dimethyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carboxamide