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6-methyl-5-[5-(1-methyl-1H-imidazol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]formamido}-N,2-dimethylpropanamide
8-(3,4,5-trimethoxyphenyl)quinoline
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]quinoxaline
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(methoxymethyl)-5-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}pyrimidine
N-{2-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
N-[1-(4-hydroxyphenyl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl}-5,6-dimethylpyrimidin-4-amine
1-{imidazo[1,2-b]pyridazin-6-yl}-4-(oxolan-3-ylmethyl)piperazine
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2-methoxyacetamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-(2-methylphenyl)piperidine-1-carboxamide
ethyl 4-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}piperidine-1-carboxylate
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-4-(benzyloxy)butan-1-one
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(adamantan-2-ylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
6-methyl-2-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)quinolin-4-ol
N-[(2S,4R,6S)-2-ethyl-6-(4-hydroxyphenyl)oxan-4-yl]acetamide
3-{1-[(2-carboxyethyl)carbamoyl]piperidin-3-yl}benzoic acid
7-(cyclopropylmethyl)-2-(3-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
(4aR,8aS)-6-[(2,5-difluorophenyl)methyl]-1-(3,3-diphenylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[(1S,5R)-6-(4-propoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(4-{[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}quinazolin-2-yl)methanol
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
3-(5-methyl-1H-pyrazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
2-[(1S,5R)-6-(1-benzofuran-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(2-oxoazepan-1-yl)propanamide
2-[2-(5-chloro-2-methoxypyridin-4-yl)-4-methylphenoxy]acetamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
5-methyl-N-(2-{[1-(pyrimidin-4-yl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
2-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
(3S,7S)-5-(dimethyl-1,3-oxazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenol
6-{methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-{[7-(3-chlorothiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methylbutanamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
N-(2-methylpropyl)-1-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-(adamantan-1-ylmethyl)-3-methoxy-1,2-dihydropyridin-2-one
8-[2-(morpholin-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]urea
2-{[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
{1-[2-(4-methylphenyl)quinoline-4-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
(1S,5R)-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyridin-2-one
2-(6-methoxypyridin-3-yl)-2-[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]acetic acid
2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide