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N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(3-methylpyridin-4-yl)methyl]amine
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-2-ol
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
1-[4-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]-4-methylpiperazine
N-ethyl-4-[5-(4-phenylbutanamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
(3S,9aR)-3-benzyl-2-methyl-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[1-(2,4-difluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-methyl-3-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
4-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
N-[(1R)-3-methyl-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butyl]acetamide
3-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
{1-[1-(methylsulfanyl)propan-2-yl]-4-(2-phenylethyl)piperidin-4-yl}methanol
2-({4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
2-ethoxy-5-(2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-3-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[(2-ethoxyphenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N1-(5-methylpyridin-2-yl)-N3-(trimethylpyrimidin-4-yl)propane-1,3-diamine
N-{[3-(cyclopentyloxy)-4-methoxyphenyl]methyl}-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-5-carboxamide
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-[2-(4-chlorophenoxy)ethyl]-N-ethyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-(2,3-difluoro-6-methoxybenzoyl)-4-(2,2-dimethoxyethyl)piperazine
3-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamido]propanamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]urea
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N,4-bis(propan-2-yl)-1,3-thiazole-2-carboxamide
4-(2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol
8-fluoro-2-({[2-(piperidin-1-yl)ethyl]amino}methyl)quinolin-4-ol
2-[6-hydroxy-4-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-1,4-diazepan-1-yl]acetic acid
2-chloro-3-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-6-methoxyphenol
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-3-[3-(1H-imidazol-1-yl)propyl]urea
(1R,2R)-N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)-2-phenylcyclopropane-1-carboxamide
N-[3-oxo-3-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propyl]acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
1-benzoyl-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
4-(pyridin-3-yl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-(3-fluoropyridin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
propan-2-yl 2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine