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N-(1,1-dioxo-1λ6-thian-4-yl)-3-(4-fluorophenyl)-N-methyl-1H-pyrazole-5-carboxamide
5-oxo-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
1-(2-{[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)amino}ethyl)piperidin-2-one
2-{[4-(propan-2-yloxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane
(2S,4R)-4-amino-1-[2-(morpholin-4-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(2-fluoro-6-methoxyphenyl)-2-(methoxymethyl)-1,3-benzoxazole
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]acetamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methanol
2-ethyl-9-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-(1,3-benzothiazol-2-yl)-2-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenol
(2S,4S)-N,N-diethyl-1-(oxan-4-yl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
(2S,3R)-3-hydroxy-2-({[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}amino)butanamide
1-(4-methylphenyl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-2-one
3-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
4-(3,4-diethoxyphenyl)-2-(oxolan-3-yl)-1H-imidazole
N-{[7-(2,2-dimethyloxane-4-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
1-(1-{4-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]phenyl}ethyl)piperidine
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-5-methyl-1,3-benzoxazole
3-(1H-pyrazol-1-ylmethyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
(2S)-N-{[1-(phenoxymethyl)cyclopropyl]methyl}pyrrolidine-2-carboxamide
2-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-4-(propan-2-yl)-1,3-thiazole
7-(4-chlorophenyl)-2-(6-hydroxypyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-methyl-2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
1-{2-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-3-ol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-{4-[4-(2,8-dimethylquinoline-4-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}propan-1-one
1-(3,5-dimethylphenyl)-4-(5-fluoro-2-methoxybenzoyl)piperazin-2-one
(4aS,7aR)-1-[4-(benzyloxy)butanoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine
4-acetamido-N,3-dimethyl-N-(quinolin-5-ylmethyl)benzamide
2-amino-4-ethyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,3-thiazole-5-carboxamide
5-[butyl(methyl)amino]-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[1-(3-methylbutyl)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
3-[(oxolan-3-yl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
N-(1,2-oxazol-3-ylmethyl)-3-[(oxolan-3-yl)sulfamoyl]benzamide
N-[2-(diethylamino)ethyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-4-methoxy-3-(morpholin-4-yl)benzamide
methyl 5-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-ethyl-1-methyl-4-[2-(2-oxopyrrolidin-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
9-methoxy-N-methyl-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-methoxy-5-methyl-N-[(3R)-piperidin-3-yl]thiophene-2-carboxamide
4-[5-(1-benzothiophen-2-ylmethyl)-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methoxy-2-phenylethan-1-one
N-(3-hydroxypropyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide