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2-methyl-5-phenyl-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
8-fluoro-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]quinoline-2-carboxamide
6-methyl-2-({[2-(pyridin-3-yl)ethyl]amino}methyl)quinolin-4-ol
N-[2-(2-fluorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
(3R,9aR)-3-benzyl-8-[(2-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,3S)-3-(2-aminoethoxy)-7-(pyridine-3-sulfonyl)-7-azaspiro[3.5]nonan-1-ol
2-[4-(8-methoxy-4-methylquinolin-2-yl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
1-[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethan-1-one
2-[5-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
5-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-phenyl-1H-imidazole-4-carboxamide
3-{1-[4-(furan-2-ylmethoxy)phenyl]-1H-imidazol-2-yl}pyridine
1'-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine
2-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]ethan-1-ol
3-[5-({[2-(4-fluorophenyl)ethyl]carbamoyl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-oxopiperidin-1-yl)propanamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-methyl-2-(phenoxymethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
5,8-dimethyl-2-({[1-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)quinolin-4-ol
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]butan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,4-dimethyl-1,2,5-oxadiazole-3-carboxamide
1-methyl-8-{[2-(methylsulfanyl)phenyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)-N-phenylpiperidine-1-carboxamide
7-(4-fluorophenyl)-2-(3-methylpyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,4-dihydropyridin-4-one
3-[4-(dimethylamino)phenyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
({[(2S,4S)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-fluoropyrrolidin-2-yl]methyl}sulfamoyl)dimethylamine
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
N-methyl-N-[1-(pyridin-3-yl)propyl]quinoxaline-5-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
(3aR,6aR)-2-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(5-methylfuran-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{[1-(2-fluorophenyl)-2,2-dimethylcyclopropyl]formamido}-N-(1,3-thiazol-2-yl)acetamide
N-({1-[(8-methylquinolin-5-yl)methyl]piperidin-3-yl}methyl)methanesulfonamide
5-{4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-[2-(1-benzofuran-2-yl)phenyl]ethan-1-amine
6-(3-fluorophenyl)-N,N-dimethylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(3-{2-[4-(3-chlorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl]morpholine
N-(2-methylquinolin-4-yl)quinoxaline-6-carboxamide
1-(4-amino-5-methylpyrimidin-2-yl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
N-[(5-methyl-1H-imidazol-4-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(2S,4S)-4-amino-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-(2-phenylethyl)piperidine
2-cyclohexyl-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
5-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-[(1-ethylpiperidin-3-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide