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3-{imidazo[1,2-a]pyridin-3-ylmethyl}-5-methoxy-3,4-dihydroquinazolin-4-one
5-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-cyclopropyl-5-[(1-phenyl-1H-pyrazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-methyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
1-(3-fluorophenyl)-5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(2-ethyl-1H-imidazol-1-yl)propanamide
1-({5-[(3S)-3-ethylmorpholine-4-carbonyl]furan-2-yl}methyl)-1H-indole
4-[4-(1-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
5-(2,4-difluorophenoxymethyl)-N-methyl-N-(quinoxalin-6-ylmethyl)-1,2-oxazole-3-carboxamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-benzyl-N-methyl-3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl 2-(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
N'-(2,4-dimethoxyphenyl)-N-[1-(1H-indol-1-yl)propan-2-yl]propanediamide
N-(furan-2-ylmethyl)-3-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propanamide
3-[3-(acetamidomethyl)phenyl]benzoic acid
1-[(4aR,8aS)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
N-(3-acetamido-4-methoxyphenyl)-7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(2-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-ethyl-4-({4-methoxy-3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)morpholine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-(2-methylprop-2-en-1-yl)-3-phenylpropanamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(pyrrolidine-3-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]propanamide
3-chloro-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[3-(4-fluorophenoxy)propyl][(2-methoxypyrimidin-5-yl)methyl]methylamine
(3S,4S)-4-(morpholin-4-yl)-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-ol
2-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-5-carboxamide
3-ethyl-8-(2-methyl-1,3-benzothiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
2-(3-methoxypropyl)-9-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(2-amino-6-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
(3S,4S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
methyl 3-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamido}propanoate
2-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-N-(propan-2-yl)acetamide
methyl 2-{4-[4-(ethylamino)pyrimidin-2-yl]-2-oxopiperazin-1-yl}acetate
2-[2-(4-fluorophenoxy)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
diethyl({[3-(3-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
3-methoxy-1-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-1,2-dihydropyridin-2-one
N-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-(4-fluorophenoxy)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
3-butyl-1-{2-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-propyl-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,4-diazepan-6-ol
2-methoxy-5-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}phenol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclobutanamine
N-[3-(dimethylamino)-1-phenylpropyl]-2,6-dimethylquinoline-4-carboxamide