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methyl 4-{[4-(2-fluorophenoxy)phenyl]carbamoyl}piperidine-1-carboxylate
2-methyl-4-[3-(4-phenyl-1,4-diazepane-1-carbonyl)phenyl]but-3-yn-2-ol
1-[1-(2-methoxybenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-[9-(3,4-difluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
6-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
2,3,5-trimethyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-5-methyl-1H-indazole
3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(cyclopropylmethyl)-5-(4-propylpyrimidine-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(1-ethyl-1H-imidazol-2-yl)piperidine
2-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1,4-diazepan-6-yl]acetic acid
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1-phenyl-1H-1,2,3-triazole
3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidine-5-carboxamide
2,3,5-trimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
5-{1-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
3-(4-methoxyphenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
5-methyl-1'-{[3-(morpholin-4-yl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-methyl-5-[5-(4-phenyl-1,3-thiazol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(1R,7S)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
9-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-benzylpiperidine-1-carbonyl)-2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-1,4-dihydropyridin-4-one
7-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)-3-(propan-2-yl)urea
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2,8-dimethylquinoline-4-carboxamide
1-[benzyl(methyl)amino]-3-[4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
ethyl 2-({3-[(furan-2-ylformamido)methyl]piperidine-1-carbonyl}amino)acetate
5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,4-dimethyl-1,3-thiazole
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
(3R,5R)-N-[2-(2,5-dimethylphenyl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[(3R,4S)-1-(2-carbamoylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-ethyl-5-methylthiophene-3-carboxamide
2-(2-methylphenyl)-1-(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1'-(1H-imidazol-2-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1-methylpiperazine-2-carboxylic acid
(1R,7S)-6-(4,4-difluoropiperidine-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
N-methyl-N-[(6-methylpyridin-2-yl)methyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-[(2-methoxyphenyl)methyl]acetamide
1-(difluoromethyl)-4-(4-methoxy-2-methylphenyl)-5-methyl-1H-pyrazole
(5-{3-[(4-methoxyphenyl)methyl]-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl}furan-2-yl)methanol
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-methylfuran-2-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}pyrimidin-4-amine
3-phenyl-5-(2-propoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-[2-(3-methoxyphenyl)-1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-(benzyloxy)-8-(2-phenoxyacetyl)-1,8-diazaspiro[4.5]decan-2-one
N-(1H-indazol-5-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide