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5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-indole
4-methyl-6-[4-({[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)piperidin-1-yl]pyrimidin-2-amine
(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
(2R)-2-amino-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(furan-2-yl)propan-1-one
2-chloro-N-[2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-(8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
2-(1-benzofuran-2-sulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
ethyl 4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-cyclohexylpropanamide
6-[2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylic acid
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
5-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(propan-2-yl)-2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-(4-methylphenyl)-2-({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)propanamide
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 2-[methyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amino]acetate
3-(4-methyl-1,3-thiazol-5-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
2,4-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidine-5-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine
4-methyl-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-6H,7H,8H-cyclopenta[g]quinolin-2-amine
(1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-2-yl)methanol
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2,3,6-trimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
(4aR,8aS)-6-cyclopropanecarbonyl-1-[3-(furan-2-yl)benzoyl]-decahydro-1,6-naphthyridine
N-(1-methoxybutan-2-yl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-benzyl-5-{3-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclobutan-1-amine
3-(4-fluorophenyl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
1-(2-methoxyacetyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(4-hydroxyphenyl)methyl]piperidine-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-5-{[methyl({[1-(propan-2-yl)pyrrolidin-3-yl]methyl})amino]methyl}benzoic acid
N-benzyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-(2-{1-[4-(4-chlorophenyl)butanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
methyl 3-benzamido-5-[(2,2-dimethylpropyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(1H-1,2,3-benzotriazole-5-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[2-oxo-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]acetamide
5-(furan-3-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenol
methyl 5-[(2-hydroxy-7-methoxyquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-4-methyl-6-phenylpyrimidine
4-[4-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]but-3-yn-1-ol
[(2S,6S)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-[3-(propan-2-yl)phenyl]urea
1-(furan-3-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-(cyclopropylmethyl)-3-[(3-methoxypiperidin-1-yl)sulfonyl]benzamide