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2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
dimethyl(3-{2-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
7-[(3-hydroxy-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(propan-2-ylsulfanyl)ethyl]acetamide
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-[3-(5-oxo-4,5-dihydro-1H-pyrazol-3-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(3-methylpyridin-4-yl)-4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4-diazepane
(2R,3S,6R)-3-(4-fluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-[(4-fluorophenyl)methyl]-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl}methanol
1-[1-(methoxymethyl)cyclobutanecarbonyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
methyl 5-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-cyclopentyl-1,1-dioxo-N-(3-phenylprop-2-yn-1-yl)-1λ6-thiane-4-carboxamide
N-(3-cyclopentylpropyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)-2-methylpyrimidine
(1R,5R)-3-(2H-1,3-benzodioxole-5-carbonyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-5-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenol
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclopropanecarboxamide
2-[(4-chlorophenyl)methyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-3-methylpiperidine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(2H-1,3-benzodioxol-4-ylmethyl)(propan-2-yl)amino]propanamide
(1R,3S)-7-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
2-(4-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
1-methyl-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(3-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-methyl-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-(5-oxo-1-propylpyrrolidin-3-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
5-ethyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1,2-oxazole-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-({7-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(2-hydroxyethyl)-2-(5-phenyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[(2,6-dichlorophenyl)methyl]-5-(2-methylpyrrolidine-1-carbonyl)pyrimidin-4-ol
1-{3-[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]propyl}pyrrolidin-2-one
3-[1-(2-hydroxybutyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]benzoic acid
N3-cyclooctyl-N5-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3-methyl-1-(2-methylpropyl)-4-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperazin-2-one
4-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-1λ6-thiane-1,1-dione
N-{1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3-methyl-1-oxobutan-2-yl}acetamide
2-[1-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]phenol