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N-{2-[4-(dimethylamino)phenyl]ethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(benzylsulfanyl)-5-(1H-imidazol-2-yl)pyrimidine
2,7,8-trimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-4-carboxamide
(2R)-2-{5-[2,5-dimethyl-1-(propan-2-yl)-1H-pyrrol-3-yl]-4-phenyl-1H-imidazol-1-yl}propanamide
N-(3-hydroxy-3-phenylpropyl)-N,2-dimethylimidazo[1,2-a]pyridine-6-carboxamide
2-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
butyl 2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
(3S,4R)-1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methylpyridine-3-carbonyl)piperidin-3-ol
5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}-1-ethyl-3-(2-phenylethyl)-1H-1,2,4-triazole
(5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2-ethoxyphenyl)methanol
6-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[4-(4-methyl-1,3-oxazole-5-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
[3-(5-{4-[1-(dimethylamino)ethyl]phenyl}-4-phenyl-1H-imidazol-1-yl)propyl]dimethylamine
{9-[(3-fluorophenyl)methyl]-3-(1H-imidazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-butyl-4-{[4-(difluoromethoxy)phenyl]methyl}-1-methylpiperazin-2-one
N-ethyl-4-hydroxy-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
6-(3-fluoro-4-methoxyphenyl)-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}imidazo[2,1-b][1,3]thiazole
3-[1-(dimethylsulfamoyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
4-{[3-(cyclopentyloxy)phenyl]methyl}piperazine-1-sulfonamide
1-methyl-2-phenyl-4-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
4-[(5-chlorofuran-2-yl)methyl]-2-(pyridin-3-yl)morpholine
4-(2,4-dioxoimidazolidin-1-yl)-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]benzamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)benzamide
1-(8-chloroquinolin-5-yl)-3-(1-methanesulfonylpiperidin-4-yl)urea
N-{4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)pyrimidine-5-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
4-(1-phenyl-1H-pyrazol-4-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
5-{[benzyl(methyl)amino]methyl}-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]-3-(furan-2-yl)propan-1-one
(1S,5R)-3-benzyl-6-[4-(1H-imidazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-chlorophenyl)-1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
1-methyl-3-[2-(methylsulfanyl)benzoyl]piperidine
3-cyclohexyl-N-(3-hydroxypropyl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
ethyl 5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 2-[(1-methylpiperidin-2-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
6-chloro-N-(3-chloro-4-propanamidophenyl)pyridine-2-carboxamide
1-(2-chlorophenyl)-3-(1-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
5-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1-cyclopentylpiperidin-2-one
2-(2-hydroxyethyl)-9-[2-(naphthalen-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[3-(oxan-4-yl)-9-[3-(1H-pyrazol-1-yl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-butyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-(thiophen-2-yl)butan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidine