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6-chloro-2-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
3-(1H-imidazol-2-ylmethyl)-5-(thiophen-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
(2S)-1-[3-(azocan-1-yl)propanoyl]pyrrolidine-2-carboxylic acid
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
methyl 2-({1-[1-(3-phenylpropyl)piperidin-4-yl]piperidin-4-yl}formamido)acetate
7-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(1H-imidazol-1-ylmethyl)-1-(3-phenoxybenzoyl)piperidine
(3aR,5R,6S,7aS)-2-(2-fluoro-4-methylbenzenesulfonyl)-octahydro-1H-isoindole-5,6-diol
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(oxan-2-ylmethoxy)acetamide
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(2-phenoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-{[({1-[ethyl(methyl)amino]cyclohexyl}methyl)amino]methyl}-1H-indol-1-yl)propanamide
{1-[3-(diphenylmethyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
2-methyl-4-(4-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}phenyl)but-3-yn-2-ol
N,N-diethyl-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-{[(3S)-1-benzylpiperidin-3-yl]amino}-N-(2-acetamidophenyl)acetamide
2-cyclopropyl-8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,8-diazaspiro[5.5]undecan-3-one
8-(2-hydroxyacetyl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4R)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-(quinolin-4-yl)piperidin-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
5-fluoro-2-[4-(trifluoromethyl)piperidin-1-yl]pyrimidin-4-ol
1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-5-oxopyrrolidine-3-carboxamide
1-(2-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(3-fluoro-4-methylphenyl)methyl]-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-(piperidin-3-yl)benzamide
1-{1-[(4-ethoxyphenyl)methyl]piperidin-3-yl}-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
8-(6-methylpyridin-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
N-butyl-N-[(2-fluorophenyl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
(1S,4S)-2-(2H-1,3-benzodioxol-5-yl)-5-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
methyl 3-[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]propanoate
6-(1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}piperidin-4-yl)-2-methyl-3,4-dihydropyrimidin-4-one
6-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}propanoic acid
8-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-(2-fluorophenyl)-4-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]piperazine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylthiophene-2-carboxamide
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidin-4-amine
[(5-ethylpyridin-2-yl)methyl]({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl})methylamine
(2S,4S)-4-amino-1-[(3,5-dichlorophenyl)methanesulfonyl]-N-ethylpyrrolidine-2-carboxamide
6-[2-(furan-2-yl)azepane-1-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(1-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile