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methyl 2-chloro-4-({[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzoate
2-ethyl-4-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyrimidine
ethyl 1-({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)piperidine-2-carboxylate
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-2-[3-(1H-pyrazol-3-yl)-1H-indazol-1-yl]acetamide
N-[(2-methoxyphenyl)methyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}cyclopropanamine
1-(2-ethoxyethyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
7-(2-aminoethyl)-N2-cyclopropyl-N4-(1-methylpiperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophene-2-carboxamide
2-({1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
N-cyclopropyl-1-{1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
1-cyclohexyl-5-(furan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
8-(6-aminopyrimidin-4-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6,8-dimethyl-2-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)quinolin-4-ol
5-[2-(2-aminoethyl)morpholine-4-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-methyl-4-(2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-4-carbonyl)piperazine
1-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-3-(hydroxymethyl)piperidin-3-ol
1-methyl-3-(2-methylpropyl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}prop-2-enamide
1-{1'-[(3-fluoro-5-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
3-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-5,6-dihydro-1,4-dioxine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(1H-imidazol-1-ylmethyl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine
N-methyl-N-(3-methylbutyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
2,3-dimethoxy-N-{[1-(quinolin-8-ylmethyl)piperidin-3-yl]methyl}benzamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1-methylpyrrolidin-2-yl)ethyl]amine
(2S,4R)-1-(furan-3-ylmethyl)-N-(propan-2-yl)-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
2-(oxolan-2-ylmethyl)-9-[(2-propoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
1,2-dimethyl-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
4-(3-ethyl-1H-pyrazole-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-methylpyridin-4-yl)-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy]-1-[4-(4-chlorophenyl)piperazin-1-yl]ethan-1-one
4-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]-1,3-thiazol-2-amine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-N-(3-methoxyphenyl)-7-azaspiro[3.5]nonane-7-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
2-cyclopropyl-6-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-benzoxazole
5-chloro-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-(3,4-difluorophenyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
(1S,5R)-6-(cyclopropylmethyl)-3-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
(2S,3R)-2-({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}amino)-3-hydroxybutanamide
N-cyclopropyl-1-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol