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4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
2-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}urea
3-[(4-cyclopentyl-3-oxopiperazin-1-yl)methyl]-7-fluoro-1,2-dihydroquinolin-2-one
N-({4-[(dimethylamino)methyl]phenyl}methyl)-2-(4-methoxyphenyl)acetamide
N-[(2-methylphenyl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1,2-oxazolidin-4-ol
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-1-(4-hydroxybutyl)-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-3-(1,2-oxazinan-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
N-[(2,5-dimethoxyphenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
2-[4-({3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)phenyl]acetic acid
2-amino-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-methylpropanamide
methyl 2-chloro-4-({[2-(dimethylamino)ethyl](ethyl)carbamoyl}amino)benzoate
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-(dimethylamino)-2-(4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
3-(4-methyl-1,3-thiazol-5-yl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)propanamide
4-benzyl-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
2-(1-ethylpyrrolidine-3-carbonyl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
N-cyclopropyl-3-[(4-fluorophenyl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-benzyl-5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
N-benzyl-3-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-N-methylpropanamide
(1S,6R)-9-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(2-hydroxybutyl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
3-phenyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidin-3-ol
3-(5-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]furan-2-carboxamide
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
1-{4-[2-(pyridin-3-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-(cyclopropylmethyl)-3-[(4-ethylpiperazin-1-yl)methyl]-3-hydroxypiperidin-2-one
N-(1-carbamoylcyclopentyl)-2-methyl-1,3-benzoxazole-6-carboxamide
3-[2-(2-methylpropanesulfonyl)ethyl]-1-(quinolin-5-yl)urea
(2S)-2-(8-methoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-3-methylbutanamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
4-{5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
(3aR,6aR)-2-(2-methoxyacetyl)-N-[2-(thiophen-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)propanamide
N2,N2,N4,N4-tetramethyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-cyclohexyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 4-{[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}butanoate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)naphthalene-2-carboxamide
6-(6-ethyl-2-methylquinoline-4-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-ethyl-N-[(4-fluorophenyl)methyl]-4-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine