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1-(2-methanesulfonylethyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine
4-cyclohexanecarbonyl-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-butanamido-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(1R,9S)-5-amino-3-(5-ethylfuran-2-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1,4-dimethylpiperidine-4-carboxamide
3-benzoyl-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1H-pyrazole-3-carboxamide
2-({4-[3-(morpholin-4-ylmethyl)phenyl]phenyl}sulfanyl)acetamide
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(2,4-difluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-cyclopropyl-2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-4-carboxamide
2-(4-fluorophenoxymethyl)-N-[(2-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
1-tert-butyl-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
2-(1-methyl-4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-2-yl)ethan-1-ol
8-[(2S)-2-amino-4-hydroxybutanoyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-2-(dimethylamino)-2-(2-methylphenyl)-N-(pyridin-4-ylmethyl)acetamide
3-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}pyridine
(2R)-2-amino-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-phenylethan-1-one
2-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}benzoic acid
N-methyl-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(3-phenylpropyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
2-(2-hydroxy-3-methylbutanoyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(2-methylpropyl)-4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-(5-{imidazo[2,1-b][1,3]thiazol-6-yl}-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl)acetic acid
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl})(pyrazin-2-ylmethyl)amine
1-(2,2-dimethylpropyl)-3-hydroxy-3-[({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]piperidin-2-one
(4aR,8aR)-2-(1-methyl-1H-pyrrole-2-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-(2-fluoro-5-methanesulfonamidophenyl)-3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]urea
N-cyclopropyl-2-{1-oxa-8-azaspiro[4.5]decan-8-yl}pyridine-4-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
6-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
1-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(2-oxopyrrolidin-3-yl)benzamide
(3S)-3-[2-(3-chloro-4-hydroxy-5-methoxyphenyl)-1H-imidazol-1-yl]azepan-2-one
N-methyl-3-[1-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-3-yl]-N-(1-methylpiperidin-4-yl)propanamide
[2-(7-chloroquinolin-4-yl)phenyl]methanol
7-(2,3-dimethoxyphenyl)-9-methoxy-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-fluorophenyl)-2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyrimidine
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
3-cyclopropyl-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4-fluorophenyl)ethyl]acetamide
1-[(2R)-pyrrolidine-2-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{[4-(4-chlorophenyl)phenyl]methyl}-3-methylpiperazin-2-one
[(1-cyclopentylpiperidin-4-yl)methyl][(4-phenyl-1,3-thiazol-2-yl)methyl](pyridin-3-ylmethyl)amine
N-ethyl-1-methyl-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-{2-[4-(dimethylamino)phenyl]acetyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
1-{3-[({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}amino)methyl]phenyl}ethan-1-one