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(2E)-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
N'-cyclopentyl-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]butanediamide
3-cyclohexyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3R,5S)-5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrrolidin-3-yl]-2-(4-methoxyphenyl)acetamide
2-methoxy-4-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyridine
4-(1H-imidazol-1-ylmethyl)-1-(1-methylazepane-2-carbonyl)piperidin-4-ol
1-[4-(3-methylphenoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
6-fluoro-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
2-cyclopentyl-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-hydroxy-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methylphenoxy)propan-1-one
5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine-2,4-diol
N-[(3R,4R)-3-hydroxy-1-(4-phenylbutanoyl)piperidin-4-yl]pyridine-4-carboxamide
7-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-6-methylpyridin-3-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1H-indole-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
(2R)-2-cyclohexyl-2-hydroxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(1S,5R)-3-[2-(ethanesulfonyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(azocane-1-carbonyl)-2-(4-fluorophenoxymethyl)pyrimidin-4-ol
ethyl 1-(cyclopent-1-ene-1-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-(furan-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]azepane
3-(oxolan-2-yl)-7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(1-benzyl-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
1-(4-acetamido-3-methoxyphenyl)-1H-indazole-3-carboxylic acid
(2S)-1-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-hydroxypropan-1-one
1-[(4-fluorophenyl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrimidine-5-carboxamide
4-(cyclopropylmethyl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
1-(2-methoxyethyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-({1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidin-3-yl}methyl)benzamide
2-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl}-1,3-thiazole
2-(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
4-[1-methyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-1-oxaspiro[4.5]decan-2-one
methyl 4-oxo-4-[6-oxo-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]butanoate
(4aR,8aR)-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}-1-(4-methylphenyl)urea
N,5-dimethyl-N-[2-(oxan-4-yl)ethyl]thiophene-2-carboxamide
3-({3-[3-(3-methylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)benzonitrile
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-(4-fluorophenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-benzyl-3-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3,5-difluorophenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-N-(5-methyl-1,2-oxazol-3-yl)acetamide
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetic acid
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
4-(4-methoxy-2-methylphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}pyrrolidine-2-carboxylate
4-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide