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7-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
3-[(3R,4S)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N2,N4-dimethyl-N2-[2-(2-methylpiperidin-1-yl)ethyl]pyrimidine-2,4-diamine
5-chloro-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-2-carboxamide
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
N-[2-(1H-indol-3-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[4-(2-butoxyacetamido)-2-chlorophenyl]propanamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-3-ylmethyl)propanamide
[1-(5-methyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperidin-4-yl]methanol
6-(benzyloxy)-1-cyclohexyl-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-2-one
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-(methoxymethyl)thiophene-2-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-hydroxy-4-methylpentan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
{[5-(4-methoxyphenyl)furan-2-yl]methyl}(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
6-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}quinoline
6-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)-2-methylpyrimidin-4-ol
1-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)-2-(propan-2-yloxy)ethan-1-one
5-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-cyclopropyl-6-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,3-benzoxazole
8-(3-fluoropyridine-4-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-{1-[4-(4-methoxyphenyl)-4-oxobutanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-cyclopropyl-5-(3-methoxyphenyl)-1H-1,2,4-triazole
N-[(2R,3R)-2-methoxy-1'-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
N-{1-[({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)carbamoyl)methyl]-1H-pyrazol-4-yl}-2H-1,3-benzodioxole-5-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(2-propoxyethyl)morpholine
2-(dimethylamino)-1-(4-ethoxypiperidin-1-yl)-2-(3-fluorophenyl)ethan-1-one
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(isoquinolin-5-ylmethyl)(methyl)(1,3-thiazol-4-ylmethyl)amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-methylpropanamide
1-(2,2-difluorocyclopropanecarbonyl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(morpholin-4-ylmethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)furan-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-[(3,4-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(trifluoromethyl)phenyl]methyl}amine
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
N-{1-[(4-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-propylmorpholine-4-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-3-[2-(methylsulfanyl)benzoyl]piperidine
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine