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4-{[(3S,4R)-4-ethoxyoxolan-3-yl]amino}-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
N-{2-[ethyl(methyl)amino]butyl}-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-(2-aminoethyl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(4-fluorophenyl)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-(3-methoxypropyl)-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
(2S,4R)-N-cyclopropyl-4-[(4-fluorophenyl)sulfanyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-4-(furan-3-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(3,4-dimethylphenyl)methyl]-4-[2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-(2-phenylethyl)pyrrolidin-1-yl]ethan-1-one
N-cyclopropyl-3-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)sulfamoyl)benzamide
5-propyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-benzyl-3-methyl-1-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-fluorophenyl)methyl]-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-ethyl-8-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-[2-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,9R)-11-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-({1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-3-yl}methyl)acetamide
methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
[(6-methylpyridin-2-yl)methyl]({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amine
4-methoxy-N-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-{2-[4-(dimethylamino)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
6-{1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)acetamide
2-(3,4-dichlorophenyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}morpholine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}piperidin-2-one
ethyl 1-{2-[4-(pyridine-2-amido)-1H-pyrazol-1-yl]acetyl}piperidine-3-carboxylate
N-ethyl-1-(piperidin-3-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-propyl-1H-pyrazole-4-carboxamide
8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(propan-2-yl)({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-1H-pyrazole-3-carboxylic acid
6-(methoxymethyl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-4-amine
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2,2,6,6-tetramethylpiperidin-4-amine
1-(4-methoxyphenyl)-3-(propan-2-yl)-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazole
6-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]quinoxaline
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1,7-dimethyl-2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-indole
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(1H-imidazol-2-ylmethyl)(2-methoxyethyl)amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(piperidin-1-ylmethyl)-N-(propan-2-yl)benzamide
7-[(2-fluorophenyl)methyl]-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3,4-dimethylbenzoyl)-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3-methylphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-3-methylpyridine-2-carboxamide