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1-[(4-ethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
2-methyl-6-(1-methyl-1H-pyrazol-4-yl)-3,4-dihydroquinazolin-4-one
1,3-dimethyl-5-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)imidazolidine-2,4-dione
6-cyclopentyl-N-[2-(4-fluorophenoxy)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carboxylate
4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
5-(4,6-dimethyl-2-oxo-2H-pyran-5-carbonyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-methyl-2-[1-(oxane-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
3-methyl-1-(3-sulfamoylphenyl)-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
(2R,3R)-3-amino-1'-[3-(trifluoromethyl)pyridin-2-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-fluoro-2-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carbonyl}quinoline
propan-2-yl 4-{[4-(pyridin-3-yloxy)phenyl]carbamoyl}piperidine-1-carboxylate
N-methyl-4-[3-(4-methylpyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(5-ethylpyridin-2-yl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
3-{1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-3-yl}benzoic acid
N-methyl-N-(2-phenylethyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
3-[5-(4-fluoro-2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
2-(dimethylamino)-4-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]pyrimidine-5-carboxamide
N-methyl-3-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
N-cyclopentyl-3-[5-(2-phenylethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
2-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
2,6-dimethyl-4-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)phenyl acetate
4-{1-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}pyridine
2-amino-N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-4-(trifluoromethyl)pyrimidine-5-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(pyridin-2-yl)ethyl]benzamide
1-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrazole-3-carboxamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine-3-carboxamide
1-[2-(dimethylamino)-4-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
methyl (2S)-2-cyclopropyl-2-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]acetate
2-(6-aminopyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
5-cyclopropyl-1-methyl-4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
(3S,4S)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}pyrrolidin-2-one
1-methyl-8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
9-(cyclopropylmethyl)-4-(3-ethoxypropanoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclobutyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
4-(4-methanesulfonylphenyl)-3-methyl-1-phenyl-1H-pyrazol-5-amine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[3-(pyridin-3-yl)propanoyl]-decahydro-2,7-naphthyridine-2-carboxamide
9-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-3,9-diazaspiro[5.6]dodecane
2-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(pyridin-2-yl)ethyl]benzamide
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
5-ethyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-1-(carboxymethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-{2-[5-(3,5-difluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[(2R)-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxobutan-2-yl]acetamide
(1S,5R)-6-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane