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2-(2-ethyl-1H-imidazol-1-yl)-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]ethan-1-one
6-cyclopentyl-N-(2-ethoxyethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-5-({3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
2-cyclopropyl-9-(5-methyl-1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
4,6-dimethyl-2-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(1-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-3-methylpyridine
(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
ethyl 4-benzyl-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-methyl-N-{1-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
methyl 5-{[(3,5-difluorophenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-chloro-4-({4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenol
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(methylsulfanyl)propan-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methylphenol
1-methyl-9-(quinoxalin-2-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-{1-[1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
1-[2-(3-fluorophenyl)ethyl]-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-6-oxopiperidine-3-carboxamide
7-(3-chlorophenyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{[benzyl(methyl)amino]methyl}-N-[(6-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
4-[(1-ethyl-1H-indol-6-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
6-fluoro-4-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
(1R,9aR)-1-({[2-(2-hydroxyethoxy)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
3-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(methoxymethyl)-N-[3-(methylsulfanyl)propyl]pyridine-2-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
1-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)piperidine-3-carbonitrile
N'-cycloheptyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]butanediamide
5-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-3,4-dihydropyrimidin-4-one
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(methylsulfanyl)pyridine-3-carboxamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-2,4,5-trifluorobenzamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(1,3-thiazol-4-yl)acetamide
1-(pyridin-3-ylmethyl)-4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
1-(1H-imidazole-2-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
14-(2,4-dimethoxy-3-methylphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N1-(6-fluoropyridin-3-yl)-N4-[(4-methoxyphenyl)methyl]piperidine-1,4-dicarboxamide
4-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}benzonitrile
[(3R,4R)-4-[(dimethylamino)methyl]-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
3-(2,6-dimethylphenoxy)-1-(2-methyloxolane-2-carbonyl)azetidine
methyl 5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
8-{3-[5-(thiophen-2-yl)furan-2-yl]propanoyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-chloro-2-hydroxy-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]benzamide