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3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
3-{[1-(3-fluorophenyl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
2-(1,3-thiazol-2-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
(2R,3R,6R)-5-(2-fluoro-6-methoxybenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2,6-dimethyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
2-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
3-methyl-1-[3-(pyridin-3-yl)propyl]-1,2-dihydroquinoxalin-2-one
N-{[1-(2-methoxyquinoline-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
6-cyclopentyl-1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-(propan-2-yl)-1,3-oxazole
ethyl 2-{4-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]morpholin-3-yl}acetate
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-(1,4-oxazepan-6-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-cyclopropyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-methyl-1H-imidazole
(4aR,7aS)-1-[2-(quinolin-6-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-oxaspiro[4.4]nonan-3-yl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
7-(5-phenyl-1,2-oxazole-3-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-(benzyloxy)-N-methyl-N-[1-(pyridin-4-yl)ethyl]butanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
2-{3-[2-amino-3-cyano-5-methyl-6-(thiophen-2-yl)pyridin-4-yl]phenoxy}acetamide
2-phenyl-N-({7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(pyridin-4-yl)piperazine
N-({1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
2-{4-methyl-6-[methyl(oxolan-3-ylmethyl)amino]pyrimidin-2-yl}phenol
2-(2H-1,3-benzodioxol-5-yl)-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(trifluoromethyl)-1H-1,3-benzodiazole
(3R,4R)-4-(azepan-1-yl)-1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-3-ol
3-methyl-1-propyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-pyrazole-4-carboxamide
2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-methoxyphenyl)-N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
4-hydroxy-1-methyl-N-[(1R,2S)-2-phenylcyclohexyl]piperidine-4-carboxamide
2-(dimethylamino)-1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
N-[(3-chloro-4-fluorophenyl)methyl]-1-ethylpiperidine-2-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-ethoxypyridine
N-cycloheptyl-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-{[7-methoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-4-methylbenzamide
5-ethyl-2-methyl-N-(piperidin-3-ylmethyl)pyrimidin-4-amine
2-[(3,4-difluorophenyl)methyl]-8-(pyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
4-(4-methylphenoxy)-1-(pyrrolidin-3-ylmethyl)piperidine
4-{1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidin-4-yl}pyridine
(1S,5R)-3-[(3,5-difluorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-ethylphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
1-{[(3R,4R)-4-(hydroxymethyl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl]methyl}piperidin-4-ol
N,N-dimethyl-1-(1H-pyrrole-2-carbonyl)azepan-4-amine