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1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
1-(2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
3-fluoro-4-[2-(4-hydroxyphenyl)-1H-imidazol-1-yl]benzoic acid
2-(2,3-difluorophenyl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-N-cycloheptylpiperidine-4-carboxamide
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyridine-2-carboxamide
4-chloro-N,N-dimethyl-5-{[methyl(quinolin-5-ylmethyl)amino]methyl}-1,3-thiazol-2-amine
3-(cyclopropylmethyl)-1-[(2-ethylpyrimidin-4-yl)methyl]piperidine-3-carboxylic acid
4-(furan-2-ylmethyl)-N-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]piperazine-1-carboxamide
4-(cyclopropylmethyl)-1-[(1,4-dimethylpiperidin-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-(2-phenoxyethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
N-(4-{[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]sulfamoyl}phenyl)acetamide
(2R)-2-{[4-(4-chlorophenoxy)piperidin-4-yl]formamido}propanamide
N2-(5-ethylpyrimidin-2-yl)-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
3-{1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(adamantan-1-ylmethyl)(methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
1-(2,2-dimethylpropyl)-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(2-methylpropyl)-1H-1,2,4-triazole
N,N-dimethyl-2-[(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-(1H-1,3-benzodiazol-1-yl)-1-(1,4-dioxane-2-carbonyl)piperidine-4-carboxylic acid
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(3-fluoro-4-methylphenyl)acetamide
(2R,6S)-4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2,6-dimethylmorpholine
2-[2-(dimethylamino)ethyl]-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-4-(4-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-dihydropyridin-2-one
3-(2H-1,3-benzodioxol-5-yl)-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[1-(3,5-dichloro-2-methoxybenzoyl)piperidin-4-yl]pyrrolidin-2-one
1-(4,4-difluoropiperidin-1-yl)-2-[4-(thiophen-3-ylmethyl)morpholin-3-yl]ethan-1-one
1-(propane-1-sulfonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
4-[2-(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]morpholine
methyl[(1-propyl-1H-imidazol-2-yl)methyl]{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclopropyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)piperidine-3-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-(2-methoxy-4-methylbenzenesulfonyl)piperidine
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(quinolin-6-ylmethyl)benzamide
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
N-cyclopropyl-3-(2-hydroxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
methyl 5-[(2-ethylpyrimidin-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methyl-1-(2-phenylethyl)urea
(3R,4R)-4-(2-methoxyethyl)-1-(6-methoxypyrimidin-4-yl)-3-methylpiperidin-4-ol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
4-(1H-indol-2-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-ethyl-1-methyl-1H-1,3-benzodiazol-7-yl}-2-methoxybenzamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
2-(2-phenyl-1H-imidazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-amine