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1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2,5-dimethoxyphenyl)ethan-1-one
4-(2-oxopyrrolidin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
N-(1-{2-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
4-methoxy-6-(pyridin-3-yl)pyrimidin-2-amine
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-N-[(2-methoxyphenyl)methyl]cyclopropanamine
4-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)-1-methylpiperidin-4-ol
ethyl({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-(3-{[(1R,3R)-3-aminocyclopentyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-methoxy-1-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-(5-{1-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)benzonitrile
5-[2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-oxoethyl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1H-1,3-benzodiazole
4-(2,1,3-benzothiadiazol-5-ylmethyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(morpholin-4-yl)propanamide
3-chloro-N-cyclopentyl-4-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
3-[5-(5-cyanopyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopentylpropanamide
3-chloro-N-cyclopentyl-4-{[1-(1H-imidazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
4-{[2-(1-cyclopentanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
(3R,4R)-1-[(6-ethoxypyridin-3-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2,3,5,6-tetramethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]benzamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidine-4-carboxylate
3-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}sulfonyl)pyridine
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(3-methoxyphenyl)ethyl]-N-methylpyridin-2-amine
N-[(1-ethylpiperidin-3-yl)methyl]-1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrazine-2-carboxamide
[(2S,4R)-1-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
2-{[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-N,N-dimethylethane-1-sulfonamide
1-{5-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]thiophen-2-yl}ethan-1-one
1-(4-{4-[(1,3-thiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
1-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-(propan-2-yloxy)acetamide
3-ethyl-1-({1-[1-(2-methylpropanoyl)piperidin-4-yl]piperidin-3-yl}methyl)urea
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridin-4-yl)propanamide
(3R,4R)-1-(2-aminopyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-(3,3-dimethylpyrrolidine-1-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-{4-oxo-4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butyl}acetamide
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
2-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-1,3-thiazole-4-carboxamide
3-[(3R,4S)-1-[(2-methylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-benzyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1,3-benzoxazole-5-carboxamide
3-[(2R,3R,6R)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
{[2-(azocan-1-yl)pyridin-3-yl]methyl}(1H-1,3-benzodiazol-2-ylmethyl)amine
3,5-dimethyl-N-{3-methyl-1-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
5-amino-4-chloro-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1H-pyrazole-3-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
2-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(furan-2-yl)-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane