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2-(thiophene-3-carbonyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
4-{3-[4-(ethoxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4-(4-{[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}phenyl)-2-methylbutan-2-ol
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 4-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]piperidine-1-carboxylate
N,N-dimethyl-2-[5-(morpholin-4-ylmethyl)pyridin-2-yl]aniline
3,5-dimethyl-1-(2-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-1H-1,2,4-triazole
(3aR,6aR)-2-cyclopentyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(2-aminopyrimidin-5-yl)-6-chloro-N-ethyl-N-(propan-2-yl)quinoline-4-carboxamide
(2S,4S)-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
2-({[1-(pyridin-4-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
3-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)propanamide
N-(1-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
2-methoxy-N-{2-[1-(oxan-4-yl)piperidin-3-yl]ethyl}pyridine-4-carboxamide
4-[(1-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]morpholine
(3-methyl-1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)methanol
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
6-(4-ethylphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3aS,6aS)-2-ethyl-5-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-({1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
1-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-(dimethylamino)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(3-methylphenyl)ethan-1-one
(2R,6R)-4-(3,5-dimethylbenzoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)-N-methylthiophene-2-carboxamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-(2H-1,3-benzodioxol-5-yl)-5-[2-(1,2-oxazolidin-2-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
4,4-diphenyl-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine
N-(1-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
4-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2,3,5-trimethyl-7-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrazolo[1,5-a]pyrimidine
2-(1-benzyl-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl)ethan-1-ol
N-cyclopentyl-1-(2-methylpropyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(cyclopropylmethyl)-5-(furan-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(6-phenoxypyridin-3-yl)-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2E)-1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(pyridin-2-yl)prop-2-en-1-one
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(4-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]urea
3-({4-[1-(3-methylfuran-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
5-chloro-4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-2-methoxyphenol
(4S,4aS,8aR)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
N-butyl-N-methyl-3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
5-propyl-1'-{thieno[2,3-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(propan-2-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole
2-{4-[(2,6-dimethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol