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3-chloro-4-{[1-(1,4-dithiepan-6-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
methyl 2-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
3-chloro-2-[(3-methoxypiperidin-1-yl)methyl]-1H-indole
(2R,6S)-2,6-dimethyl-4-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
9-methoxy-3-(oxolane-2-carbonyl)-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-fluoropiperidine
[(5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-3-yl)methyl]dimethylamine
1-methyl-N-(2-oxoazepan-3-yl)-1H-1,3-benzodiazole-5-carboxamide
3-(2,3-dihydro-1H-isoindol-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
2-(1,3-benzoxazol-2-yl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)methylamine
1-(pyrimidin-2-yl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane
5-(1-cyclopropanecarbonylpyrrolidin-2-yl)-N-(2-methoxypyridin-3-yl)thiophene-2-carboxamide
2-[3-methoxy-5-(trifluoromethyl)phenyl]-N,N-dimethylpyridine-3-carboxamide
3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
N-{4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-4-oxobutyl}acetamide
1-(1,3-thiazol-4-ylmethyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-(3-hydroxypiperidin-1-yl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
9-(cyclopropylmethyl)-4-(2,5-dimethylfuran-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-fluorophenyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
4-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
4-(2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)morpholine
4-methyl-3-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-4H-1,2,4-triazole
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(pyridin-3-yl)pentyl]urea
N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-cyclohexyl-1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
3-ethyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(propan-2-yl)acetamide
1-{5-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-2-methylphenyl}imidazolidin-2-one
3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[(3S,4R)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{4-[(2,5-difluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-methyl-5-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-thiazole
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
6-[({5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}amino)methyl]-1,4-oxazepan-6-ol
2-(azepan-1-yl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
3-[2-(dimethylamino)ethyl]-8-fluoro-3,4-dihydroquinazolin-4-one
(4aS,8aR)-6-[(3-methyl-1H-indol-2-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[3-(oxolan-2-yl)propyl]benzamide
6-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-1H-pyrrolo[2,3-b]pyridine
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-methylpropyl)piperidine
6-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one