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3-[(2-fluorophenyl)formamido]-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]propanamide
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
8-(2,3-dihydro-1H-indene-1-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(3aS,7aR)-5-methyl-2-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}-N-[(3-methyloxetan-3-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
1,3-dimethyl-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2R)-1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
3-(morpholine-4-carbonyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-8-methoxy-4-methylquinoline
2-(4-methyl-6-{[1-(pyrazin-2-yl)piperidin-3-yl]amino}pyrimidin-2-yl)phenol
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[2-(pyridin-2-yl)ethyl]amine
N-methyl-3-propyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-{5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-cyclopentyl-1H-1,2,4-triazol-1-yl}acetic acid
3-cyclohexyl-N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}propanamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-N-[2-(ethylsulfanyl)ethyl]cyclohexanamine
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(3,4-dimethoxyphenyl)methyl]methylamine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
4-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2,3-thiadiazole
2-({2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
4-methoxy-N-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
2-(2,3,4-trimethoxyphenyl)benzonitrile
1-{2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-3,5-dimethyl-1H-1,2,4-triazole
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
[(5-methylthiophen-2-yl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
4-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}benzoic acid
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-methoxybutan-1-one
7-methyl-4-(2-methylpiperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
3-[(methylsulfanyl)methyl]-5-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
2-methoxy-4-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carbonitrile
3-methyl-3-phenyl-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
2,5-dimethyl-N-[3-(morpholin-4-yl)propyl]-1,3-thiazole-4-carboxamide
N-butyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(pyridin-4-ylmethyl)acetamide
N-ethyl-N-(oxolan-2-ylmethyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2,5-dimethoxy-N-methylbenzamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}dimethylamine
N,2,5,7-tetramethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-ethyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-indole-5-carboxamide
(2S,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
N-{2-[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
5-chloro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,3-dihydro-1H-indole-2-carboxamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-[(1S)-1-acetamidoethyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,3,5,6-tetramethylbenzamide
8-[2-(2,3,4-trifluorophenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid