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2-oxo-6-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}-1,2-dihydropyridine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(3,4-dimethylbenzenesulfonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-{2-methyl-5-[3-(3-methylphenyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
1-(dimethylamino)-2-{4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(4-chloro-1H-pyrazol-1-yl)ethan-1-one
2-[(1S)-1-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl]-3-methylpyridine
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-chloro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-methyl-2-[3-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyridine
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[1-(thian-4-yl)piperidin-4-yl]propan-1-one
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(4-chlorophenyl)-1-benzofuran-2-carboxamide
3-[3-(2,4-dimethoxyphenyl)phenyl]-1H-pyrazole
(2S,4R)-N-ethyl-1-methyl-4-(2-{[(2-methylphenyl)methyl]sulfanyl}acetamido)pyrrolidine-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-2-methylfuran-3-carboxamide
2-[5-cyclopropyl-4-(4-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2,5-dimethylthiophen-3-yl)pyrimidine
1-[(4aR,8aR)-4a-hydroxy-7-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-(1-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
(2-methylpropyl)({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-2-ylmethyl)amine
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-propoxypiperidine
N2-(2-methoxyethyl)-N4-(pyridin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
1-(2-chlorophenyl)-4-[2-(pyridin-2-ylsulfanyl)propanoyl]piperazin-2-one
N-[3-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
5-(1-benzofuran-2-yl)-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
N-(thiolan-3-yl)quinoxaline-5-carboxamide
4-({5-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
2-(2H-1,3-benzodioxol-5-yl)-1-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
6-(morpholin-4-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenol
(3S,4R)-4-methyl-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine-3,4-diol
2-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-methyl-1,6-naphthyridine-3-carboxamide
3-[5-(3-ethoxybenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(3R,5S)-N3-[(4-methoxyphenyl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
5-{[4-(acetamidomethyl)piperidin-1-yl]methyl}-2-hydroxybenzoic acid
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[4-(2-oxopyrrolidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(1-methanesulfonylpiperidin-4-yl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(2-methylprop-2-en-1-yl)amino]pyridine-3-carboxamide
N-(butan-2-yl)-2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
2-(difluoromethoxy)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)benzamide
6-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[2-methoxy-4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
4-(cyclopropylmethyl)-1-(5-methylthiophene-2-carbonyl)-1,4-diazepan-5-one
(2S)-3-(4-hydroxyphenyl)-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanoic acid
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide