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2-ethyl-N-methyl-N-(quinolin-5-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-acetamido-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
N-tert-butyl-2-(4-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}phenoxy)acetamide
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methoxyethan-1-one
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-phenylpiperidine
4-{[propyl(pyridin-4-ylmethyl)amino]methyl}benzene-1,2-diol
1-(carbamoylmethyl)-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1-{[1-(2,3-dihydro-1H-indene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
ethyl 2-{1-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]piperidin-2-yl}acetate
methyl 1-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
4-(4-chlorophenoxy)-N-ethyl-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
N3-[2-(2-methoxyphenyl)ethyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
dimethyl[(4-methyl-5-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
2-(3-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
2-[3-(azepan-1-ylmethyl)phenyl]-6-(4-hydroxyphenyl)-3,4-dihydropyrimidin-4-one
(1R,2S)-2-[4-(2-methoxyphenyl)-3-oxopiperazine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
2-(thiophen-2-yl)-5-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyrimidine
N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1H-pyrazol-1-yl)benzamide
2-methyl-5-[4-({[4-(methylamino)pyrimidin-2-yl]amino}methyl)piperidin-1-yl]-2,3-dihydropyridazin-3-one
8-fluoro-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}quinoline
N3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-({5-[(2-methoxynaphthalen-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-({[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}methyl)-4-hydroxyquinoline-6-carboxamide
4-(3-methyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole
4-(6-fluoro-1H-1,3-benzodiazol-2-yl)phenol
3-methyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-(2-chlorophenyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}phenol
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(pyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]thiolan-3-amine
(2S,4S)-4-amino-N-ethyl-1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
1-cyclopropyl-5-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrrolidine-3-carboxamide
N-(2-methyl-5-{[(5-oxo-1-propylpyrrolidin-3-yl)carbamoyl]amino}phenyl)propanamide
2-benzyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-amine
N-[(1S,2R)-2-aminocyclobutyl]-3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaene-9-sulfonamide
5-(furan-2-yl)-3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
6-[3-(hydroxymethyl)piperidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(1H-pyrazol-3-ylmethyl)amine
(2S,4R)-4-amino-N-(propan-2-yl)-1-[(5-propylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(thiophen-3-yl)acetamide
1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
ethyl 4-{[(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)carbamoyl]amino}piperidine-1-carboxylate
(3R,5R)-5-(morpholine-4-carbonyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide