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7-(2H-1,3-benzodioxole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[(2S,4S)-1-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-4-fluoropyrrolidin-2-yl]methyl}acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
7-[2-(4-benzylpiperazin-1-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
5-[2-(2-chlorophenoxymethyl)pyrimidin-4-yl]-2-ethoxybenzoic acid
1-[2-methoxy-5-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]pyridin-3-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
6-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
(2S,4R)-4-amino-N-ethyl-1-(4-methoxy-2-methylbenzoyl)pyrrolidine-2-carboxamide
2-{[4-(2-methyl-5-propylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
1-(2-methoxyphenyl)-4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]piperazine
1-{2-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2-phenoxyethan-1-one
2-(2-hydroxyethyl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-acetyl-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,2,4-trimethyl-1H-pyrrole-3-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-[(5-chlorothiophen-2-yl)methyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
4-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-2-[(4-fluorophenyl)methyl]morpholine
N-[2-(diethylamino)ethyl]-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(4-amino-3-hydroxybutanoyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
2-methyl-4-{4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
N-cyclohexyl-3-{[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]formamido}propanamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
(3S,4R)-1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-one
1-[(4-chlorophenyl)methyl]-1-(3-hydroxypropyl)-3-(3-methoxy-4-methylphenyl)urea
2-(2-methoxyethyl)-8-(5-methyl-1,3,4-oxadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-(4-methoxyphenoxy)-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
6-(1,5-dimethyl-1H-indole-2-carbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
N-cyclopentyl-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-(3-phenylprop-2-yn-1-yl)acetamide
4-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}-N-methylbenzene-1-sulfonamide
3-(1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-2-yl)ethan-1-one
8-methoxy-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-(3-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-1H-indol-1-yl)acetamide
2-cyclopropyl-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
8-(dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(4-chloro-1-ethyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
(2R,3R,6R)-5-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)({5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
(4S)-4-(methoxymethyl)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3,3-dimethylpiperidin-4-ol
{1-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]piperidin-2-yl}methanol
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
2-(3-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
7-(cyclobutylmethyl)-2-(3-hydroxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
(2-chloro-6-fluorophenyl)[4-(3-phenyl-1,2-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol