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4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(cyclopropylmethyl)pyrimidine
3-{[5-(2,3-dihydro-1H-inden-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(5-methyl-1,3-thiazol-2-yl)benzamide
(2R,3R)-3-{[2-(pyrazin-2-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-cyclopropyl-3-[5-(5-methoxyfuran-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
2,8-dimethyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
4-{[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzonitrile
(2S,4R)-1-(cyclohexylmethyl)-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(1,3-dimethyl-1H-pyrazol-4-yl)acetamide
5-[(pyrimidin-2-ylsulfanyl)methyl]-N-[1-(thiophen-2-yl)propan-2-yl]furan-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
2-[(3-methoxyphenyl)amino]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}butanamide
3-(1H-1,3-benzodiazol-2-yl)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
3-{[1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-fluorobenzamide
1-[4-(oxan-2-ylmethoxy)phenyl]-3-{2-[(pyridin-3-yl)amino]ethyl}urea
3-(1H-imidazol-2-yl)-N-(2-oxoazepan-3-yl)benzamide
4-[(2,5-difluorophenyl)methyl]-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-N-[(4-methoxyphenyl)methyl]-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{[2-(2-aminoethyl)quinazolin-4-yl]amino}butan-2-ol
(2-methoxyethyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(propan-2-yl)amine
2-butyl-8-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-(piperidin-3-yl)benzamide
2-[(4-chlorophenyl)sulfanyl]-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
6-[(diethylamino)methyl]-N-[2-(1H-imidazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-acetamidoacetyl)piperidine-3-carboxylate
N-(4-methylphenyl)-4-{[4-(morpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-[1-(3-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-(methylsulfanyl)propanamide
N,N-dimethyl-3-(3-methylthiophene-2-carbonyl)piperidine-1-sulfonamide
1-{2-[3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-(3,5-dimethyl-4-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(3-methoxyphenyl)methyl]-3-[1-(pyrimidin-5-ylmethyl)piperidin-3-yl]propanamide
2-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-1H-1,3-benzodiazole
2-(4-fluorophenyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
(2H-1,3-benzodioxol-4-ylmethyl)[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
2-(3-fluoro-5-methoxyphenyl)-2-[4-(2-hydroxyphenyl)piperazin-1-yl]acetic acid
3-{1-[5-(2-fluoro-3-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
1-[(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)methyl]-3,5-dimethyl-1H-pyrazole
2-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
N-cyclohexyl-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide