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[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-1H-indol-3-yl)methyl](pyridin-3-ylmethyl)amine
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(thiophen-3-yl)acetamide
2-{4-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-6-methylpyrimidin-2-yl}phenol
4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
3-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
N,N-diethyl-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}aniline
8-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(1S)-2,3-dihydro-1H-inden-1-yl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclohexyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)propanamide
2-{5-[(2S)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
4-fluorophenyl (7S,9aR)-7-[(4-methoxyphenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(2E)-3-(4-fluorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-en-1-one
2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]naphthalen-1-ol
[(3S,5R)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-({methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-8-ol
2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxylic acid
2-[4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]-1,3-benzothiazole
N-methyl-N-[2-(morpholin-4-yl)propyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-methoxy-3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
1-ethyl-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(4-methoxyphenyl)-N,2,2-trimethylcyclopropane-1-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
N-(2-methoxyethyl)-5-methyl-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}thieno[2,3-d]pyrimidin-4-amine
2-{[(5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
2-(2-hydroxyethyl)-3-oxo-N-{3-[(trifluoromethyl)sulfanyl]phenyl}piperazine-1-carboxamide
(4aR,7aS)-1-(2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-4-(2-methoxyethyl)piperazine
methyl 6-({[1-(1H-imidazol-1-yl)butan-2-yl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
1-[7-(3-chlorophenyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
N-[1-({[(3-methoxyphenyl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
1-[2-(4-methylpiperazine-1-carbonyl)piperazin-1-yl]-5-phenylpentan-1-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-(4-propanoylphenoxy)acetamide
4-{[1-(2-oxo-1,2-dihydroquinoline-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-(2,6-dimethylpyridin-4-yl)-4-(2-methyl-1-benzofuran-5-carbonyl)piperazine
2-methyl-1-{4-[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidin-1-yl}propan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-decahydroisoquinoline
7-(propan-2-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
N-{2-[({6,7-dimethoxy-2-[(4-methylphenyl)methoxy]quinolin-3-yl}methyl)amino]ethyl}acetamide
{5-[1-(2,3-dihydro-1H-inden-4-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
ethyl 2-[4-(5-acetylpyridin-2-yl)piperazin-1-yl]acetate
(2S)-2,6-diamino-1-[3-(3-methylphenoxy)azetidin-1-yl]hexan-1-one