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5-methoxy-1-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-indole-2-carboxamide
4-benzyl-3-ethyl-1-[2-(methylamino)pyridine-3-carbonyl]-1,4-diazepan-5-one
3-(4-methanesulfonylphenyl)-5-methylpyridin-2-amine
1-(2-methylphenyl)-4-{2-[2-(trifluoromethyl)phenyl]acetyl}piperazin-2-one
(4aS,8aS)-2-cyclohexyl-7-(6-methoxypyrimidin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyrimidin-4-amine
2-{6-[(propan-2-yl)amino]pyridazin-3-yl}benzoic acid
3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2,1-benzoxazole
7-methyl-2-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
5-(3,4-dimethylphenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
1-methyl-9-[(2-propoxyphenyl)methyl]-1,4,9-triazaspiro[5.5]undecan-5-one
5-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
(2S,4R)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-(furan-2-amido)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N,2,5,6-tetramethyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine
2-benzyl-N-[2-(1H-indol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
1-(4-methylphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(1H-pyrazol-1-yl)benzamide
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-1-{3-[2-methyl-6-(trifluoromethyl)pyridin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-1-one
1-methyl-2-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-indole
4-(1-cyclopentanecarbonylpyrrolidin-3-yl)-1-(2-phenylethyl)piperidine
6-[(2,6-difluorophenyl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-methyl-3-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)quinoxaline
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(2-methylphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
2-cyclopentyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenylacetamide
1-(2,6-difluorophenyl)-3-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]urea
6-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[2-(dimethylamino)ethyl]-5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-1-[(3-chlorophenyl)methyl]-1H-1,2,4-triazole
3-{2-[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(1S,5R)-3-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-methanesulfonamidophenyl)-4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carboxamide
N-[2-(diethylamino)ethyl]-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
methyl 4-(5-chloro-2-{[2-(methylsulfanyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N,N-dimethyl-3-{4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}aniline
1-{2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
methyl 6-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-2-(cyclopropylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
11-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
3-[4-fluoro-3-(hydroxymethyl)phenyl]-5-(thiomorpholine-4-sulfonyl)benzoic acid
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]propanamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(1H-indole-6-carbonyl)piperidin-3-yl]propanamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
6,7-difluoro-3-[(1-methylpiperidin-2-yl)methyl]-3,4-dihydroquinazolin-4-one
N-cyclobutyl-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-1,4-diazepan-5-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-[5-(6-methoxynaphthalen-2-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,2-diol
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]imidazo[1,2-a]pyridine-2-carboxamide