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N-cyclopropyl-4-methoxy-3-({1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}oxy)benzamide
methyl 3-(furan-2-ylmethyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-4-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-amine
N-(2-methoxyethyl)-3,4,7-trimethyl-N-(1-methylpiperidin-4-yl)-1H-indole-2-carboxamide
3-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}phenol
4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]phenol
5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
(1R,5S,6S)-6-({4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
2-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}-5-ethylpyrimidine
1-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(methylsulfanyl)-N-(pyridin-3-ylmethyl)acetamide
8-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({1-[(3-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}methyl)morpholine
1-(3-{5-[(dimethylamino)methyl]pyridin-2-yl}phenyl)ethan-1-one
2-[(1S,5R)-6-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
2-(dimethylamino)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
3-hydroxy-3-{[(oxan-4-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
1-{4-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
4-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-one
1-(1,4-dioxan-2-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,6-dimethylquinoline
4-(3,4-diethoxyphenyl)-2-(1-methyl-1H-imidazol-5-yl)-1H-imidazole
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-ethylpyrimidin-2-amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
3-(6-phenylpyridazin-3-yl)-3,9-diazaspiro[5.6]dodecan-10-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
5-(2-chlorophenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}furan-2-carboxamide
3-cyclopropyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1,2-oxazole-5-carboxamide
4-{5-[(3-methoxy-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}morpholine
N-{[3-(oxolan-3-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}cyclopropanamine
N-({1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-methylfuran-2-carboxamide
methyl 4-({[2-(azocan-1-yl)pyridin-3-yl]methyl}carbamoyl)butanoate
1-(2-methoxyethyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
1-(2-methoxy-4-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
1-(adamantan-1-yl)-4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-chlorophenol
1-(2-{[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]methyl}morpholin-4-yl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}propanamide
1-[2-(4-aminoazepan-1-yl)-2-oxoethyl]-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyrrolidin-1-yl)piperidine
(3aR,6aR)-N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
3-[(3R,4S)-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(thian-4-yl)piperidine
3-(4-methyl-1H-pyrazol-5-yl)-1-(naphthalene-2-sulfonyl)piperidine