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2-(adamantan-1-yl)-1-[4-(pyridin-4-yloxy)piperidin-1-yl]ethan-1-one
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)propanamide
8-(2,2-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
1-[(4-chlorophenyl)methyl]-5-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
1-[(3-fluorophenyl)methyl]-4-[(6-methyl-2-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
2-methoxy-5-({[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]carbamoyl}amino)benzamide
(4aR,7aS)-1-{2-[2-(pyrrolidin-1-yl)phenoxy]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-fluoro-N-[1-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-4-carbonitrile
(4aS,8aR)-6-(5-methoxy-1H-indazole-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{[2-methyl-4-(4-methylphenyl)piperazin-1-yl]methyl}-2-propylpyrimidine
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2-(thiophen-2-yl)azetidine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
3-propoxy-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
4-(hydroxymethyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-ol
7-methyl-3-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)thiomorpholine
3-(pyridin-3-yl)-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
3-[1-(methoxymethyl)cyclopentyl]-1-[3-(1H-pyrazol-1-yl)phenyl]urea
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1,2-dihydropyridin-2-one
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-(3-methoxyphenyl)azetidine
N-[2-(3-chlorophenyl)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-methyl-6-(pyridin-4-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(2-fluorophenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N'-{2-[(2-fluorophenyl)carbamoyl]ethyl}-N-[2-(methylsulfanyl)phenyl]butanediamide
3-({2-[1-(2-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2,8-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-4-carboxamide
5-{1-[3-(3,4-difluorophenyl)propanoyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
4-(2-cyclohexylpyrimidin-5-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(4-chlorophenyl)methyl]-8-(2-hydroxyethyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-7-methoxy-4-methylquinoline
(3aS,6aS)-2-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[1-(3-chloro-4-methoxybenzoyl)piperidin-2-yl]ethyl}acetamide
3-[(4aR,7aS)-4-[2-(4-hydroxyphenyl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(pyridin-3-ylmethyl)-4-{[3-({1-[4-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine
4-(2-chloro-3-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
2-amino-4-[2-methoxy-5-oxo-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl]-5H,6H,7H,8H,9H-cyclohepta[b]pyridine-3-carbonitrile
6-fluoro-2-oxo-N-[4-(pyridin-2-yl)butyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-(4-chlorobenzenesulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
2-(dimethyl-1,3-thiazol-5-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-methyl-2-(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)-1H-imidazole
2-(carbamoylamino)-N-[(3R,4S)-1-(cyclobutylmethyl)-4-propylpyrrolidin-3-yl]acetamide
4-(5-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(propan-2-yloxy)ethyl]benzamide
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide