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N-benzyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-({3-[(2S)-4-methyl-2-(propan-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-fluoro-4-(quinolin-3-yl)benzene-1-sulfonamide
3-ethoxy-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1R,2R,6S,7S)-4-[(3,4-dimethoxypyridin-2-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-(5-acetyl-2-ethoxyphenyl)-3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
8-[(4-methoxypyridin-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-methoxyacetyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
2-(5-{[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]methyl}furan-2-yl)benzonitrile
N-(3-ethylphenyl)-4-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-4-oxobutanamide
4-[(4-chlorophenyl)methanesulfonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
5-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-cyclopentylpiperazine
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-propylpyrrolidin-3-amine
2-{1-[(2-tert-butyl-5-carbamoylfuran-3-yl)methyl]pyrrolidin-3-yl}benzoic acid
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-phenylpiperidine
N-(3-chlorophenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
3-{[(1S)-1-carbamoyl-2-hydroxyethyl]sulfamoyl}-N-cyclobutylbenzamide
3-{3-[2-(methylamino)ethoxy]phenyl}phenol
N-{1-[(1-methyl-1H-imidazol-2-yl)methyl]azepan-3-yl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-[4-(4-{2-[3-({methyl[(5-oxopyrrolidin-2-yl)methyl]amino}methyl)phenoxy]ethyl}piperazine-1-carbonyl)phenyl]pyrrolidin-2-one
1-{[5-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2,4-dimethylphenyl]methyl}-1H-1,2,4-triazole
8-acetyl-2-{[5-(methylcarbamoyl)furan-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-benzyl-3-[1-(2-chloropyridine-4-carbonyl)piperidin-4-yl]-N-methylpropanamide
1-(2-cycloheptylethyl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
methyl[(2-methyl-1H-imidazol-4-yl)methyl][(1-phenylpyrrolidin-3-yl)methyl]amine
methyl (1S,3R,3aR,6aS)-3-(2,2-dimethylpropyl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
9-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-oxa-9-azaspiro[5.5]undecane
5-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
N-(2-cyclooctylethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
3-(4-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
ethyl 5-[({1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)methyl]furan-2-carboxylate
2,2,2-trifluoro-1-[4-(quinolin-5-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,3-dihydroxypropyl)-N-methyl-1H-pyrazole-3-carboxamide
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(4aR,8aR)-2-[3-(methylsulfanyl)propyl]-7-(pyrimidin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
4-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
1-[3-(azepan-1-yl)propyl]-3-(1-benzyl-1H-pyrazol-5-yl)-1-methylurea
3-{2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
(3S,5S)-1-benzyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(3-phenoxyphenyl)methyl]pyrrolidin-3-amine