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N-[(3R,4S)-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-4-propylpyrrolidin-3-yl]acetamide
N-ethyl-N-[2-(2-methylphenoxy)ethyl]-2-(morpholin-2-yl)acetamide
4-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-1-ethyl-1,2-dihydropyridin-2-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-methylbut-2-en-1-one
2-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propane-1,3-diol
7-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidine
5-methyl-1'-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(4-methylpentyl)morpholin-4-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
4-[5-(5-ethyl-1H-pyrrol-2-yl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl]benzamide
1-[1-(pyridine-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(2R)-1-(3-{[3-hydroxy-2-(hydroxymethyl)-2-methylpropyl]carbamoyl}benzenesulfonyl)pyrrolidine-2-carboxamide
6-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2,4-dimethylpyridine-3-carbonitrile
6-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-ethyl-4-methyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,3-oxazole-5-carboxamide
1-[2-methoxy-4-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-{5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(naphthalen-1-yl)-1H-1,2,4-triazol-3-yl}acetamide
2-(4-methylpentyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]morpholine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-methyl-4-(4-methylphenyl)piperazine
3-ethyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[2-(prop-2-en-1-yloxy)phenyl]urea
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
ethyl 5-{[(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazol-4-yl)formamido]methyl}furan-2-carboxylate
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-thiazole-4-carboxamide
4-{[4-(4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-propyl-1,2-oxazole-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-[5-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)thiophen-2-yl]prop-2-yn-1-ol
N,N-dimethyl-2-({[5-(trifluoromethyl)pyridin-2-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
8-[1-(piperidin-1-yl)cyclohexanecarbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(4-{2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-4-yl}-1H-1,2,3-triazol-1-yl)methyl]-1λ6-thiolane-1,1-dione
6-ethyl-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
(1S,5R)-1,3,3-trimethyl-6-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-6-azabicyclo[3.2.1]octane
2-(4,5-dichloro-1H-imidazol-1-yl)-N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]acetamide
N-(2-hydroxybutyl)-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-cyclohexyl-1-(4,7-dimethylquinazolin-2-yl)azepan-4-amine
2-[4-(dimethylamino)azepane-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-methyl-4-(4-methylpiperazin-1-yl)-N-[1-(thiophen-2-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[5-(1H-1,3-benzodiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
5-[({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
1-methyl-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
2-{[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
N-[(3R,4S)-1-[(3E)-4-methylhex-3-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-[5-(furan-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
3-(1H-1,3-benzodiazol-1-yl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one